PDB entry 4yjr
View 4yjr on RCSB PDB site
Description: SYK kinase domain in complex with inhibitor GTC000225
Class: transferase
Keywords: syk, non-receptor tyrosine kinase, spleen tyrosine kinase, transferase, phosphorylation, transferase-transferase inhibitor complex
Deposited on
2015-03-03, released
2015-09-30
The last revision prior to the SCOPe 2.07 freeze date was dated
2015-09-30, with a file datestamp of
2015-09-25.
Experiment type: XRAY
Resolution: 1.32 Å
R-factor: N/A
AEROSPACI score: 0.58
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Tyrosine-protein kinase SYK
Species: Homo sapiens [TaxId:9606]
Gene: SYK
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4yjra_ - Heterogens: 4DJ, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4yjrA (A:)
peeirpkevyldrklltledkelgsgnfgtvkkgyyqmkkvvktvavkilkneandpalk
dellaeanvmqqldnpyivrmigiceaeswmlvmemaelgplnkylqqnrhvkdkniiel
vhqvsmgmkyleesnfvhrdlaarnvllvtqhyakisdfglskalradenyykaqthgkw
pvkwyapecinyykfssksdvwsfgvlmweafsygqkpyrgmkgsevtamlekgermgcp
agcpremydlmnlcwtydvenrpgfaavelrlrnyyydvvn
Sequence, based on observed residues (ATOM records): (download)
>4yjrA (A:)
yldrklltledkelgtvkkgyyqmkkvvktvavkilkneandpalkdellaeanvmqqld
npyivrmigiceaeswmlvmemaelgplnkylqqnrhvkdkniielvhqvsmgmkylees
nfvhrdlaarnvllvtqhyakisdfglskalradenyykaqthgkwpvkwyapecinyyk
fssksdvwsfgvlmweafsygqkpyrgmkgsevtamlekgermgcpagcpremydlmnlc
wtydvenrpgfaavelrlrnyyydv