PDB entry 4xp3

View 4xp3 on RCSB PDB site
Description: Crystal structure of ERK2 in complex with an inhibitor
Class: transferase
Keywords: SERINE/THREONINE-PROTEIN KINASE, transferase
Deposited on 2015-01-16, released 2015-08-12
The last revision prior to the SCOPe 2.05 freeze date was dated 2015-08-12, with a file datestamp of 2015-08-07.
Experiment type: XRAY
Resolution: 1.78 Å
R-factor: N/A
AEROSPACI score: 0.38 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Mitogen-activated protein kinase 1
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Mapk1, Erk2, Mapk, Prkm1
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.05: d4xp3a_
  • Heterogens: DX4, SO4, DMS, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >4xp3A (A:)
    gpemvrgqvfdvgprytnlsyigegaygmvcsaydnlnkvrvaikkispfehqtycqrtl
    reikillrfrheniigindiiraptieqmkdvyivqdlmetdlykllktqhlsndhicyf
    lyqilrglkyihsanvlhrdlkpsnlllnttcdlkicdfglarvadpdhdhtgflteyva
    trwyrapeimlnskgytksidiwsvgcilaemlsnrpifpgkhyldqlnhilgilgspsq
    edlnciinlkarnyllslphknkvpwnrlfpnadskaldlldkmltfnphkrieveqala
    hpyleqyydpsdepiaeapfkfdmelddlpkeklkelifeetarfqpgyrs
    

    Sequence, based on observed residues (ATOM records): (download)
    >4xp3A (A:)
    gpemvrgqvfdvgprytnlsyigegaygmvcsaydnlnkvrvaikkispfehqtycqrtl
    reikillrfrheniigindiiraptieqmkdvyivqdlmetdlykllktqhlsndhicyf
    lyqilrglkyihsanvlhrdlkpsnlllnttcdlkicdfglarvadpdhdhtgflteyva
    trwyrapeimlnskgytksidiwsvgcilaemlsnrpifpgkhyldqlnhilgilgspsq
    edlnciinlkarnyllslphknkvpwnrlfpnadskaldlldkmltfnphkrieveqala
    hpyleqyydpsdepiaeapfkflpkeklkelifeetarfqp