PDB entry 4x6n
View 4x6n on RCSB PDB site
Description: FACTOR XIA IN COMPLEX WITH THE INHIBITOR 1-{(1S)-1-[4-(3-amino-1H-indazol-6-yl)-5-chloro-1H-imidazol-2-yl]-2-phenylethyl}-3-[5-chloro-2-(1H-tetrazol-1-yl)benzyl]urea
Class: hydrolase/hydrolase inhibitor
Keywords: SERINE PROTEASE, BLOOD COAGULATION FACTOR, PROTEIN INHIBITOR COMPLEX, hydrolase-hydrolase inhibitor complex
Deposited on
2014-12-08, released
2015-02-18
The last revision prior to the SCOPe 2.06 freeze date was dated
2015-04-01, with a file datestamp of
2015-03-27.
Experiment type: XRAY
Resolution: 2.1 Å
R-factor: N/A
AEROSPACI score: 0.29
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: coagulation factor xi, light chain
Species: Homo sapiens [TaxId:9606]
Gene: F11
Database cross-references and differences (RAF-indexed):
- Uniprot P03951 (0-237)
- engineered mutation (103)
- engineered mutation (105)
Domains in SCOPe 2.06: d4x6na_ - Chain 'H':
Compound: cleaved peptide
Species: Homo sapiens [TaxId:9606]
Gene: F11
Database cross-references and differences (RAF-indexed):
- Heterogens: 3Y5, SO4, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4x6nA (A:)
ivggtasvrgewpwqvtlhttsptqrhlcggsiignqwiltaahcfygvespkilrvysg
ilnqseikedtsffgvqeiiihdqykmaesgydiallklettvgygdsqrpiclpskgdr
nviytdcwvtgwgyrklrdkiqntlqkakiplvtneecqkryrghkithkmicagyregg
kdackgdsggplsckhnevwhlvgitswgegcaqrerpgvytnvveyvdwilektqavhh
hhhh
Sequence, based on observed residues (ATOM records): (download)
>4x6nA (A:)
ivggtasvrgewpwqvtlhttsptqrhlcggsiignqwiltaahcfygvespkilrvysg
ilnqseikedtsffgvqeiiihdqykmaesgydiallklettvgygdsqrpiclpskgdr
nviytdcwvtgwgyrklrdkiqntlqkakiplvtneecqkryrghkithkmicagyregg
kdackgdsggplsckhnevwhlvgitswgegcaqrerpgvytnvveyvdwilektqav
- Chain 'H':
No sequence available.