PDB entry 4x1f
View 4x1f on RCSB PDB site
Description: Crystal structure of the hPXR-LBD in complex with the synthetic estrogen 17alpha-ethinylestradiol
Class: gene regulation
Keywords: nuclear receptor, hormone receptor, pregnane X receptor, estrogen, gene regulation
Deposited on
2014-11-24, released
2015-09-09
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-07-04, with a file datestamp of
2018-06-29.
Experiment type: XRAY
Resolution: 2 Å
R-factor: N/A
AEROSPACI score: 0.32
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Nuclear receptor subfamily 1 group I member 2
Species: Homo sapiens [TaxId:9606]
Gene: NR1I2, PXR
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4x1fa_ - Heterogens: 3WF, MPD, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4x1fA (A:)
mkkghhhhhhgsertgtqplgvqglteeqrmmirelmdaqmktfdttfshfknfrlpgvl
ssgcelpeslqapsreeaakwsqvrkdlcslkvslqlrgedgsvwnykppadsggkeifs
llphmadmstymfkgiisfakvisyfrdlpiedqisllkgaafelcqlrfntvfnaetgt
wecgrlsycledtaggfqqlllepmlkfhymlkklqlheeeyvlmqaislfspdrpgvlq
hrvvdqlqeqfaitlksyiecnrpqpahrflflkimamltelrsinaqhtqrllriqdih
pfatplmqelfgitgs
Sequence, based on observed residues (ATOM records): (download)
>4x1fA (A:)
glteeqrmmirelmdaqmktfdttfshfknfrlpgveaakwsqvrkdlcslkvslqlrge
dgsvwnykppadsggkeifsllphmadmstymfkgiisfakvisyfrdlpiedqisllkg
aafelcqlrfntvfnaetgtwecgrlsycledqqlllepmlkfhymlkklqlheeeyvlm
qaislfspdrpgvlqhrvvdqlqeqfaitlksyiecnrpqpahrflflkimamltelrsi
naqhtqrllriqdihpfatplmqelfgitgs