PDB entry 4wkq
View 4wkq on RCSB PDB site
Description: 1.85 angstrom structure of EGFR kinase domain with gefitinib
Class: transferase/transferase inhibitor
Keywords: inhibitor, complex, kinase, epidermal growth factor receptor, TRANSFERASE, transferase-transferase inhibitor complex
Deposited on
2014-10-03, released
2014-11-05
The last revision prior to the SCOPe 2.05 freeze date was dated
2014-11-05, with a file datestamp of
2014-10-31.
Experiment type: XRAY
Resolution: 1.85 Å
R-factor: 0.196
AEROSPACI score: 0.41
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Epidermal growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: EGFR, ERBB, ERBB1, HER1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d4wkqa_ - Heterogens: IRE, NA, MES, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4wkqA (A:)
gamgeapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelreats
pkankeildeayvmasvdnphvcrllgicltstvqlitqlmpfgclldyvrehkdnigsq
yllnwcvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfglakllgaeekeyhae
ggkvpikwmalesilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekger
lpqppictidvymimvkcwmidadsrpkfreliiefskmardpqrylviqgdermhlpsp
tdsnfyralmdeedmddvvdadeylipqqg
Sequence, based on observed residues (ATOM records): (download)
>4wkqA (A:)
amgeapnqallrilketefkkikvlgsgtvykglwipegekvkipvaikespkankeild
eayvmasvdnphvcrllgicltstvqlitqlmpfgclldyvrehkdnigsqyllnwcvqi
akgmnyledrrlvhrdlaarnvlvktpqhvkitdfglakllgaeekeyhaeggkvpikwm
alesilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekgerlpqppicti
dvymimvkcwmidadsrpkfreliiefskmardpqrylviqgdmddvvdadeylipq