PDB entry 4uxq
View 4uxq on RCSB PDB site
Description: FGFR4 in complex with Ponatinib
Class: transferase
Keywords: transferase, kinase dfg-out fgfr inhibitor complex
Deposited on
2014-08-27, released
2014-12-03
The last revision prior to the SCOPe 2.05 freeze date was dated
2014-12-17, with a file datestamp of
2014-12-12.
Experiment type: XRAY
Resolution: 1.85 Å
R-factor: 0.2048
AEROSPACI score: 0.4
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Fibroblast growth factor receptor 4
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d4uxqa_ - Heterogens: SO4, 0LI, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4uxqA (A:)
gsaglvsldlpldplwefprdrlvlgkplgegafgqvvraeafgmdparpdqastvavkm
lkdnasdkdladlvsemevmkligrhkniinllgvctqegplyvivecaakgnlreflra
rrppgpdlspdgprssegplsfpvlvscayqvargmqylesrkcihrdlaarnvlvtedn
vmkiadfglargvhhidyykktsngrlpvkwmapealfdrvythqsdvwsfgillweift
lggspypgipveelfsllreghrmdrpphcppelyglmrecwhaapsqrptfkqlveald
kvllavsee
Sequence, based on observed residues (ATOM records): (download)
>4uxqA (A:)
ldlpldplwefprdrlvlgkplgegafgqvvraeafgmdparpdqastvavkmlkdnasd
kdladlvsemevmkligrhkniinllgvctqegplyvivecaakgnlreflrarrppgpl
sfpvlvscayqvargmqylesrkcihrdlaarnvlvtednvmkiadfglargvhhidyyk
ktsngrlpvkwmapealfdrvythqsdvwsfgillweiftlggspypgipveelfsllre
ghrmdrpphcppelyglmrecwhaapsqrptfkqlvealdkvllav