PDB entry 4u7z
View 4u7z on RCSB PDB site
Description: Mitogen-Activated Protein Kinase Kinase (MEK1) bound to G805
Class: TRANSFERASE/TRANSFERASE Inhibitor
Keywords: Kinase, inhibitor, Complex
Deposited on
2014-07-31, released
2014-09-24
The last revision prior to the SCOPe 2.08 freeze date was dated
2014-10-08, with a file datestamp of
2014-10-03.
Experiment type: XRAY
Resolution: 2.81 Å
R-factor: 0.163
AEROSPACI score: 0.25
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Dual specificity mitogen-activated protein kinase kinase 1
Species: Homo sapiens [TaxId:9606]
Gene: MAP2K1, MEK1, PRKMK1
Database cross-references and differences (RAF-indexed):
- Uniprot Q02750 (1-End)
- initiating methionine (0)
Domains in SCOPe 2.08: d4u7za1, d4u7za2 - Heterogens: MG, 3EW, ANP, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4u7zA (A:)
melkdddfekiselgagnggvvfkvshkpsglvmarklihleikpairnqiirelqvlhe
cnspyivgfygafysdgeisicmehmdggsldqvlkkagripeqilgkvsiavikgltyl
rekhkimhrdvkpsnilvnsrgeiklcdfgvsgqlidsmansfvgtrsymsperlqgthy
svqsdiwsmglslvemavgrypipppdakelelmfgcqvegdaaetpprprtpgrplssy
gmdsrppmaifelldyivnepppklpsgvfslefqdfvnkcliknpaeradlkqlmvhaf
ikrsdaeevdfagwlcstiglnqpstpthaagvlqhhhhhh
Sequence, based on observed residues (ATOM records): (download)
>4u7zA (A:)
melkdddfekiselgagnggvvfkvshkpsglvmarklihleikpairnqiirelqvlhe
cnspyivgfygafysdgeisicmehmdggsldqvlkkagripeqilgkvsiavikgltyl
rekhkimhrdvkpsnilvnsrgeiklcdfgvsgqlidsmansvgtrsymsperlqgthys
vqsdiwsmglslvemavgrypipppdakelelmfppmaifelldyivnepppklpsgvfs
lefqdfvnkcliknpaeradlkqlmvhafikrsdaeevdfagwlcstigln