PDB entry 4u79
View 4u79 on RCSB PDB site
Description: Crystal structure of human JNK3 in complex with a benzenesulfonamide inhibitor.
Class: transferase/transferase inhibitor
Keywords: Transferase
Deposited on
2014-07-30, released
2014-10-08
The last revision prior to the SCOPe 2.05 freeze date was dated
2014-10-08, with a file datestamp of
2014-10-03.
Experiment type: XRAY
Resolution: 2.23 Å
R-factor: 0.218
AEROSPACI score: 0.29
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 10
Species: Homo sapiens [TaxId:9606]
Gene: MAPK10, JNK3, JNK3A, PRKM10, SAPK1B
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d4u79a_ - Heterogens: 3EL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4u79A (A:)
mskskvdnqfysvevgdstftvlkryqnlkpigsgaqgivcaaydavldrnvaikklsrp
fqnqthakrayrelvlmkcvnhkniisllnvftpqktleefqdvylvmelmdanlcqviq
meldhermsyllyqmlcgikhlhsagiihrdlkpsnivvksdctlkildfglartagtsf
mmtpyvvtryyrapevilgmgykenvdiwsvgcimgemvrhkilfpgrdyidqwnkvieq
lgtpcpefmkklqptvrnyvenrpkyagltfpklfpdslfpadsehnklkasqardllsk
mlvidpakrisvddalqhpyinvwydpaeveapppqiydkqlderehtieewkeliykev
mnse
Sequence, based on observed residues (ATOM records): (download)
>4u79A (A:)
vdnqfysvevgdstftvlkryqnlkpigsggivcaaydavldrnvaikklsrpfqnqtha
krayrelvlmkcvnhkniisllnvftpqktleefqdvylvmelmdanlcqviqmeldher
msyllyqmlcgikhlhsagiihrdlkpsnivvksdctlkildfglartvtryyrapevil
gmgykenvdiwsvgcimgemvrhkilfpgrdyidqwnkvieqlgtpcpefmkklqptvrn
yvenrpkyagltfpklfpdslfpadsehnklkasqardllskmlvidpakrisvddalqh
pyinvwydpaeveapplderehtieewkeliykevmn