PDB entry 4qyf
View 4qyf on RCSB PDB site
Description: CHK1 kinase domain in complex with aminopyrazine compound 13
Class: Transferase/Transferase Inhibitor
Keywords: protein kinase, phosphotransfer catalyst, Transferase-Transferase Inhibitor complex
Deposited on
2014-07-24, released
2014-12-17
The last revision prior to the SCOPe 2.05 freeze date was dated
2014-12-17, with a file datestamp of
2014-12-12.
Experiment type: XRAY
Resolution: 2.15 Å
R-factor: 0.171
AEROSPACI score: 0.35
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase Chk1
Species: Homo sapiens [TaxId:9606]
Gene: CHEK1, CHK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d4qyfa_ - Heterogens: 3DV, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4qyfA (A:)
mavpfvedwdlvqtlgegaygevqlavnrvteeavavkivdmkravdcpenikkeicink
mlnhenvvkfyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvy
lhgigithrdikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellk
rrefhaepvdvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsapla
llhkilvenpsaritipdikkdrwynkplkkgakrprvtsggvsespsgghhhhhhhh
Sequence, based on observed residues (ATOM records): (download)
>4qyfA (A:)
vpfvedwdlvqtlgegaygevqlavnrvteeavavkivdmknikkeicinkmlnhenvvk
fyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvylhgigithr
dikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkrrefhaepv
dvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplallhkilven
psaritipdikkdrwynkplkkgaprvts