PDB entry 4qxi
View 4qxi on RCSB PDB site
Description: Crystal structure of human AR complexed with NADP+ and AK198
Class: Oxidoreductase
Keywords: TIM barrel, Aldose reductase, oxidoreductase, diabetes, Halogenated compound, Cytosolic
Deposited on
2014-07-21, released
2015-07-22
The last revision prior to the SCOPe 2.06 freeze date was dated
2015-07-22, with a file datestamp of
2015-07-17.
Experiment type: XRAY
Resolution: 0.87 Å
R-factor: N/A
AEROSPACI score: 0.97
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: aldose reductase
Species: Homo sapiens [TaxId:9606]
Gene: AKR1B1, ALDR1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d4qxia_ - Heterogens: NAP, I98, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4qxiA (A:)
masrillnngakmpilglgtwksppgqvteavkvaidvgyrhidcahvyqnenevgvaiq
eklreqvvkreelfivsklwctyhekglvkgacqktlsdlkldyldlylihwptgfkpgk
effpldesgnvvpsdtnildtwaameelvdeglvkaigisnfnhlqvemilnkpglkykp
avnqiechpyltqekliqycqskgivvtaysplgspdrpwakpedpslledprikaiaak
hnkttaqvlirfpmqrnlvvipksvtperiaenfkvfdfelssqdmttllsynrnwrvca
llsctshkdypfheef
Sequence, based on observed residues (ATOM records): (download)
>4qxiA (A:)
masrillnngakmpilglgtwksppgqvteavkvaidvgyrhidcahvyqnenevgvaiq
eklreqvvkreelfivsklwctyhekglvkgacqktlsdlkldyldlylihwptgfkpgk
effpldesgnvvpsdtnildtwaameelvdeglvkaigisnfnhlqvemilnkpglkykp
avnqiechpyltqekliqycqskgivvtaysplgspdrpwakpedpslledprikaiaak
hnkttaqvlirfpmqrnlvvipksvtperiaenfkvfdfelssqdmttllsynrnwrvca
llsctshkdypfhe