PDB entry 4qmq

View 4qmq on RCSB PDB site
Description: MST3 in complex with CP-673451
Class: Transferase/transferase inhibitor
Keywords: PROTEIN KINASE, MST3, STK24, STERILE 20-LIKE KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-TRANSFERASE, Transferase-transferase inhibitor complex
Deposited on 2014-06-16, released 2015-07-01
The last revision prior to the SCOPe 2.08 freeze date was dated 2016-07-13, with a file datestamp of 2016-07-08.
Experiment type: XRAY
Resolution: 1.77 Å
R-factor: N/A
AEROSPACI score: 0.38 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Serine/threonine-protein kinase 24
    Species: Homo sapiens [TaxId:9606]
    Gene: MST3, STK24, STK3
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d4qmqa_
  • Heterogens: 34U, EDO, PEG, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >4qmqA (A:)
    gplgsefmahspvqsglpgmqnlkadpeelftklekigkgsfgevfkgidnrtqkvvaik
    iidleeaedeiediqqeitvlsqcdspyvtkyygsylkdtklwiimeylgggsaldllep
    gpldetqiatilreilkgldylhsekkihrdikaanvllsehgevkladfgvagqltdtq
    ikrntfvgtpfwmapevikqsaydskadiwslgitaielargepphselhpmkvlflipk
    nnpptlegnyskplkefveaclnkepsfrptakellkhkfilrnakktsyltelidrykr
    wkaeqshdds
    

    Sequence, based on observed residues (ATOM records): (download)
    >4qmqA (A:)
    glpgmqnlkadpeelftklekigkgsfgevfkgidnrtqkvvaikiidleeaedeiediq
    qeitvlsqcdspyvtkyygsylkdtklwiimeylgggsaldllepgpldetqiatilrei
    lkgldylhsekkihrdikaanvllsehgevkladfgvagqltdtqikrntfvgtpfwmap
    evikqsaydskadiwslgitaielargepphselhpmkvlflipknnpptlegnyskplk
    efveaclnkepsfrptakellkhkfilrnakktsyltelidrykrwkaeq