PDB entry 4pd4
View 4pd4 on RCSB PDB site
Description: Structural analysis of atovaquone-inhibited cytochrome bc1 complex reveals the molecular basis of antimalarial drug action
Class: oxidoreductase/inhibitor
Keywords: Cytochrome bc1 complex, Membrane protein complex, antimalarial drug, inhibitor, OXIDOREDUCTASE-INHIBITOR complex
Deposited on
2014-04-17, released
2014-06-11
The last revision prior to the SCOPe 2.07 freeze date was dated
2017-11-22, with a file datestamp of
2017-11-17.
Experiment type: XRAY
Resolution: 3.04 Å
R-factor: N/A
AEROSPACI score: 0.11
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Cytochrome b-c1 complex subunit 1, mitochondrial
Species: Saccharomyces cerevisiae (strain ATCC 204508 / S288c) [TaxId:559292]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4pd4a1, d4pd4a2 - Chain 'B':
Compound: Cytochrome b-c1 complex subunit 2, mitochondrial
Species: Saccharomyces cerevisiae (strain ATCC 204508 / S288c) [TaxId:559292]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4pd4b1, d4pd4b2 - Chain 'C':
Compound: cytochrome b
Species: Saccharomyces cerevisiae (strain ATCC 204508 / S288c) [TaxId:559292]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4pd4c1, d4pd4c2 - Chain 'D':
Compound: Cytochrome c1, heme protein, mitochondrial
Species: Saccharomyces cerevisiae (strain ATCC 204508 / S288c) [TaxId:559292]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4pd4d1, d4pd4d2 - Chain 'E':
Compound: Cytochrome b-c1 complex subunit Rieske, mitochondrial
Species: Saccharomyces cerevisiae (strain ATCC 204508 / S288c) [TaxId:559292]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4pd4e1, d4pd4e2 - Chain 'F':
Compound: Cytochrome b-c1 complex subunit 6
Species: Saccharomyces cerevisiae (strain ATCC 204508 / S288c) [TaxId:559292]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4pd4f_ - Chain 'G':
Compound: Cytochrome b-c1 complex subunit 7
Species: Saccharomyces cerevisiae (strain ATCC 204508 / S288c) [TaxId:559292]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4pd4g_ - Chain 'H':
Compound: Cytochrome b-c1 complex subunit 8
Species: Saccharomyces cerevisiae (strain ATCC 204508 / S288c) [TaxId:559292]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4pd4h_ - Chain 'I':
Compound: Cytochrome b-c1 complex subunit 9
Species: Saccharomyces cerevisiae (strain ATCC 204508 / S288c) [TaxId:559292]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4pd4i_ - Chain 'J':
Compound: Igh protein
Species: Mus musculus [TaxId:10090]
Gene: IGH
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4pd4j_ - Chain 'K':
Compound: Ig kappa chain V-V region HP 124E1
Species: Mus musculus [TaxId:10090]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4pd4k_ - Heterogens: UMQ, 3PH, HEM, AOQ, 3PE, UQ6, FES
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>4pd4A (A:)
aevtqlsngivvatehnpsahtasvgvvfgsgaanenpynngvsnlwkniflskensava
akeglalssnisrdfqsyivsslpgstdksldflnqsfiqqkanllsssnfeatkksvlk
qvqdfedndhpnrvlehlhstafqntplslptrgtleslenlvvadlesfannhflnsna
vvvgtgnikhedlvnsiesknlslqtgtkpvlkkkaaflgsevrlrddtlpkawislave
gepvnspnyfvaklaaqifgsynafepasrlqgiklldniqeyqlcdnfnhfslsykdsg
lwgfstatrnvtmiddlihftlkqwnrltisvtdteveraksllklqlgqlyesgnpvnd
anllgaevlikgsklslgeafkkidaitvkdvkawagkrlwdqdiaiagtgqieglldym
rirsdmsmmrw
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>4pd4B (B:)
ltvsardaptkistlavkvhggsryatkdgvahllnrfnfqntntrsalklvresellgg
tfkstldreyitlkatflkddlpyyvnaladvlyktafkpheltesvlpaarydyavaeq
cpvksaedqlyaitfrkglgnpllydgvervslqdikdfadkvytkenlevsgenvvead
lkrfvdesllstlpagkslvsksepkfflgeenrvrfigdsvaaigipvnkaslaqyevl
anyltsalselsglissakldkftdgglftlfvrdqdsavvssnikkivadlkkgkdlsp
ainytklknavqnesvsspielnfdavkdfklgkfnyvavgdvsnlpyldel
- Chain 'C':
Sequence; same for both SEQRES and ATOM records: (download)
>4pd4C (C:)
mafrksnvylslvnsyiidspqpssinywwnmgsllglclviqivtgifmamhyssniel
afssvehimrdvhngyilrylhangasfffmvmfmhmakglyygsyrsprvtlwnvgvii
filtiataflgyccvygqmshwgatvitnlfsaipfvgndivswlwggfsvsnptiqrff
alhylvpfiiaamvimhlmalhihgssnplgitgnldripmhsyfifkdlvtvflfmlil
alfvfyspntlghpdnyipgnplvtpasivpewyllpfyailrsipdkllgvitmfaail
vllvlpftdrsvvrgntfkvlskffffifvfnfvllgqigachvevpyvlmgqiatfiyf
ayfliivpvistienvlfyigrvnk
- Chain 'D':
Sequence; same for both SEQRES and ATOM records: (download)
>4pd4D (D:)
mtaaehglhapayawshngpfetfdhasirrgyqvyrevcaachsldrvawrtlvgvsht
neevrnmaeefeyddepdeqgnpkkrpgklsdyipgpypneqaaraanqgalppdlsliv
karhggcdyifslltgypdeppagvalppgsnynpyfpggsiamarvlfddmveyedgtp
attsqmakdvttflnwcaepehderkrlglktviilsslyllsiwvkkfkwagiktrkfv
fnppkprk
- Chain 'E':
Sequence; same for both SEQRES and ATOM records: (download)
>4pd4E (E:)
kstyrtpnfddvlkenndadkgrsyayfmvgamgllssagakstvetfissmtatadvla
makvevnlaaiplgknvvvkwqgkpvfirhrtpheiqeansvdmsalkdpqtdadrvkdp
qwlimlgicthlgcvpigeagdfggwfcpchgshydisgrirkgpaplnleipayefdgd
kvivg
- Chain 'F':
Sequence; same for both SEQRES and ATOM records: (download)
>4pd4F (F:)
vtdqledlrehfknteegkalvhhyeecaervkiqqqqpgyadlehkedcveeffhlqhy
ldtataprlfdklk
- Chain 'G':
Sequence; same for both SEQRES and ATOM records: (download)
>4pd4G (G:)
pqsftsiarigdyilkspvlsklcvpvanqfinlagykklglkfddliaeenpimqtalr
rlpedesyarayriirahqtelthhllprnewikaqedvpyllpyileaeaaakekdeld
nievsk
- Chain 'H':
Sequence; same for both SEQRES and ATOM records: (download)
>4pd4H (H:)
gppsgktymgwwghmggpkqkgitsyavspyaqkplqgifhnavfnsfrrfksqflyvli
pagiywywwkngneyneflyskagreelervnv
- Chain 'I':
Sequence; same for both SEQRES and ATOM records: (download)
>4pd4I (I:)
sfsslyktffkrnavfvgtifagafvfqtvfdtaitswyenhnkgklwkdvkariaa
- Chain 'J':
Sequence; same for both SEQRES and ATOM records: (download)
>4pd4J (J:)
evklqesgaglvqpsqslsltcsvtgysitsgyywnwirlfpgnklewvgyisnvgdnny
npslkdrlsitrdtsknqfflklnsvttedtatyycarseyysvtgyamdywgqgttvtv
ssawrhp
- Chain 'K':
Sequence; same for both SEQRES and ATOM records: (download)
>4pd4K (K:)
dieltqtpvslaaslgdrvtiscrasqdinnflnwyqqkpdgtiklliyytsrlhagvps
rfsgsgsgtdysltisnlepediatyfcqhhikfpwtfgagtkleik