PDB entry 4nj3
View 4nj3 on RCSB PDB site
Description: Modulating the interaction between CDK2 and Cyclin A with a Quinoline-based inhibitor
Class: transferase/transferase inhibitor
Keywords: CELL CYCLE, INHIBITION, CYCLIN-DEPENDENT KINASE, CANCER, ATP-BINDING, CELL DIVISION,MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, transferase-transferase inhibitor complex
Deposited on
2013-11-08, released
2013-11-27
The last revision prior to the SCOPe 2.03 freeze date was dated
2013-11-27, with a file datestamp of
2013-11-22.
Experiment type: XRAY
Resolution: 1.85 Å
R-factor: 0.184
AEROSPACI score: 0.41
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cyclin-dependent kinase 2
Species: Homo sapiens [TaxId:9606]
Gene: CDK2, CDKN2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d4nj3a_ - Heterogens: 2KD, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4nj3A (A:)
menfqkvekigegtygvvykarnkltgevvalkkirldtetegvpstaireisllkelnh
pnivklldvihtenklylvfeflhqdlkkfmdasaltgiplpliksylfqllqglafchs
hrvlhrdlkpqnllintegaikladfglarafgvpvrtythevvtlwyrapeillgckyy
stavdiwslgcifaemvtrralfpgdseidqlfrifrtlgtpdevvwpgvtsmpdykpsf
pkwarqdfskvvppldedgrsllsqmlhydpnkrisakaalahpffqdvtkpvphlrl
Sequence, based on observed residues (ATOM records): (download)
>4nj3A (A:)
menfqkvekigegtygvvykarnkltgevvalkkirldpstaireisllkelnhpnivkl
ldvihtenklylvfeflhqdlkkfmdasaltgiplpliksylfqllqglafchshrvlhr
dlkpqnllintegaikladfglarevvtlwyrapeillgckyystavdiwslgcifaemv
trralfpgdseidqlfrifrtlgtpdevvwpgvtsmpdykpsfpkwarqdfskvvpplde
dgrsllsqmlhydpnkrisakaalahpffqdvtkpvphlrl