PDB entry 4n70
View 4n70 on RCSB PDB site
Description: Pim1 Complexed with a pyridylcarboxamide
Class: transferase/transferase inhibitor
Keywords: kinase, phosphorylation, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2013-10-14, released
2013-11-06
The last revision prior to the SCOPe 2.08 freeze date was dated
2014-07-02, with a file datestamp of
2014-06-27.
Experiment type: XRAY
Resolution: 2.1 Å
R-factor: 0.169
AEROSPACI score: 0.37
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase pim-1
Species: Homo sapiens [TaxId:9606]
Gene: PIM1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4n70a_ - Heterogens: 2HX, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4n70A (A:)
mahhhhhhlevlfqgpllskinslahlraapcndlhatklapgkekeplesqyqvgpllg
sggfgsvysgirvsdnlpvaikhvekdrisdwgelpngtrvpmevvllkkvssgfsgvir
lldwferpdsfvlilerpepvqdlfdfitergalqeelarsffwqvleavrhchncgvlh
rdikdenilidlnrgelklidfgsgallkdtvytdfdgtrvysppewiryhryhgrsaav
wslgillydmvcgdipfehdeeiirgqvffrqrvssecqhlirwclalrpsdrptfeeiq
nhpwmqdvllpqetaeihlhslspgpsk
Sequence, based on observed residues (ATOM records): (download)
>4n70A (A:)
eplesqyqvgpllgsggfgsvysgirvsdnlpvaikhvekdrisdwgelpngtrvpmevv
llkkvssgfsgvirlldwferpdsfvlilerpepvqdlfdfitergalqeelarsffwqv
leavrhchncgvlhrdikdenilidlnrgelklidfgsgallkdtvytdfdgtrvysppe
wiryhryhgrsaavwslgillydmvcgdipfehdeeiirgqvffrqrvssecqhlirwcl
alrpsdrptfeeiqnhpwmqdvllpqetaeihlhs