PDB entry 4mzs
View 4mzs on RCSB PDB site
Description: Mouse cathepsin s with covalent ligand (3S,4S)-1-[(2-CHLOROPHENYL)SULFONYL]-N-[(2E)-2-IMINOETHYL]-4-(MORPHOLIN-4-YLCARBONYL)PYRROLIDINE-3-CARBOXAMIDE
Class: hydrolase/hydrolase inhibitor
Keywords: HYDROLASE, CYSTEINE PROTEASE, hydrolase-hydrolase inhibitor complex
Deposited on
2013-09-30, released
2014-08-20
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-11-15, with a file datestamp of
2017-11-10.
Experiment type: XRAY
Resolution: 1.85 Å
R-factor: N/A
AEROSPACI score: 0.34
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cathepsin S
Species: Mus musculus [TaxId:10090]
Gene: Ctss, Cats
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4mzsa_ - Chain 'B':
Compound: cathepsin S
Species: Mus musculus [TaxId:10090]
Gene: Ctss, Cats
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4mzsb_ - Heterogens: 2EV, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4mzsA (A:)
rsysnrtlpdtvdwrekgcvtevkyqgscgacwafsavgalegqlklktgklislsaqnl
vdcsneekygnkgcgggymteafqyiidnggieadasypykamdekchynsknraatcsr
yiqlpfgdedalkeavatkgpvsvgidashssfffyksgvyddpsctgnvnhgvlvvgyg
tldgkdywlvknswglnfgdqgyirmarnnknhcgiasycsypei
Sequence, based on observed residues (ATOM records): (download)
>4mzsA (A:)
lpdtvdwrekgcvtevkyqgscgacwafsavgalegqlklktgklislsaqnlvdcsnee
kygnkgcgggymteafqyiidnggieadasypykamdekchynsknraatcsryiqlpfg
dedalkeavatkgpvsvgidashssfffyksgvyddpsctgnvnhgvlvvgygtldgkdy
wlvknswglnfgdqgyirmarnnknhcgiasycsypei
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4mzsB (B:)
rsysnrtlpdtvdwrekgcvtevkyqgscgacwafsavgalegqlklktgklislsaqnl
vdcsneekygnkgcgggymteafqyiidnggieadasypykamdekchynsknraatcsr
yiqlpfgdedalkeavatkgpvsvgidashssfffyksgvyddpsctgnvnhgvlvvgyg
tldgkdywlvknswglnfgdqgyirmarnnknhcgiasycsypei
Sequence, based on observed residues (ATOM records): (download)
>4mzsB (B:)
lpdtvdwrekgcvtevkyqgscgacwafsavgalegqlklktgklislsaqnlvdcsnee
kygnkgcgggymteafqyiidnggieadasypykamdekchynsknraatcsryiqlpfg
dedalkeavatkgpvsvgidashssfffyksgvyddpsctgnvnhgvlvvgygtldgkdy
wlvknswglnfgdqgyirmarnnknhcgiasycsypei