PDB entry 4lpb
View 4lpb on RCSB PDB site
Description: Crystal structure of a topoisomerase ATPase inhibitor
Class: isomerase/isomerase inhibitor
Keywords: protein-inhibitor complex, ATP binding, structure-based drug design, antimicrobial, virtual screen, ATP binding domain, ISOMERASE-ISOMERASE INHIBITOR complex
Deposited on
2013-07-15, released
2013-10-30
The last revision prior to the SCOPe 2.08 freeze date was dated
2014-01-15, with a file datestamp of
2014-01-10.
Experiment type: XRAY
Resolution: 1.75 Å
R-factor: 0.195
AEROSPACI score: 0.44
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Topoisomerase IV subunit B
Species: Streptococcus pneumoniae [TaxId:171101]
Gene: parE, spr0756
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4lpba_ - Heterogens: 1YP, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4lpbA (A:)
mskkeininnynddaiqvlegldavrkrpgmyigstdgaglhhlvweivdnavdealsgf
gdridvtinkdgsltvqdhgrgmptgmhamgiptveviftilhaggkfgqggyktsgglh
gvgssvvnalsswleveitrdgavykqrfenggkpvttlkkigtalksktgtkvtfmpda
tifsttdfkyntiserlnesafllknvtlsltdkrtdeaiefhyen
Sequence, based on observed residues (ATOM records): (download)
>4lpbA (A:)
qvlegldavrkrpgmyigstdgaglhhlvweivdnavdealsgfgdridvtinkdgsltv
qdhgrgmptgmhamgiptveviftilhavgssvvnalsswleveitrdgavykqrfengg
kpvttlkkigtalksktgtkvtfmpdatifsttdfkyntiserlnesafllknvtlsltd
krtdeaiefhyen