PDB entry 4l7r
View 4l7r on RCSB PDB site
Description: Human artd3 (parp3) - catalytic domain in complex with inhibitor ME0400
Class: transferase/transferase inhibitor
Keywords: DIPHTHERIA TOXIN LIKE ADP-RIBOSE TRANSFERASE, TRANSFERASE, ADP-RIBOSYLATION, transferase-transferase inhibitor complex
Deposited on
2013-06-14, released
2014-02-19
The last revision prior to the SCOPe 2.03 freeze date was dated
2014-02-19, with a file datestamp of
2014-02-14.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: 0.179
AEROSPACI score: 0.34
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Poly [ADP-ribose] polymerase 3
Species: Homo sapiens [TaxId:9606]
Gene: ADPRT3, ADPRTL3, PARP3
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d4l7ra1, d4l7ra2 - Heterogens: M00, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4l7rA (A:)
smkrvqpcsldpatqklitnifskemfkntmalmdldvkkmplgklskqqiargfealea
leealkgptdggqsleelsshfytviphnfghsqpppinspellqakkdmllvladiela
qalqavseqektveevphpldrdyqllkcqlqlldsgapeykviqtyleqtgsnhrcptl
qhiwkvnqegeedrfqahsklgnrkllwhgtnmavvaailtsglrimphsggrvgkgiyf
asensksagyvigmkcgahhvgymflgevalgrehhintdnpslkspppgfdsviarght
epdptqdteleldgqqvvvpqgqpvpcpefssstfsqseyliyqesqcrlryllevh
Sequence, based on observed residues (ATOM records): (download)
>4l7rA (A:)
mkrvqpcsldpatqklitnifskemfkntmalmdldvkkmplgklskqqiargfealeal
eealkdggqsleelsshfytviphnfghsqpppinspellqakkdmllvladielaqalq
avseqektveevphpldrdyqllkcqlqlldsgapeykviqtyleqtgsnhrcptlqhiw
kvnqegeedrfqahsklgnrkllwhgtnmavvaailtsglrimphsggrvgkgiyfasen
sksagyvigmkcgahhvgymflgevalgrehhintdnpslkspppgfdsviarghtepdp
tqdteleldgqqvvvpqgqpvpcpefssstfsqseyliyqesqcrlryllevh