PDB entry 4l6z
View 4l6z on RCSB PDB site
Description: Human artd3 (parp3) - catalytic domain in complex with inhibitor STO1168
Class: transferase/transferase inhibitor
Keywords: DIPHTHERIA TOXIN LIKE ADP-RIBOSE TRANSFERASE, TRANSFERASE, ADP-RIBOSYLATION, transferase-transferase inhibitor complex
Deposited on
2013-06-13, released
2014-02-19
The last revision prior to the SCOPe 2.08 freeze date was dated
2014-02-19, with a file datestamp of
2014-02-14.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.164
AEROSPACI score: 0.4
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Poly [ADP-ribose] polymerase 3
Species: Homo sapiens [TaxId:9606]
Gene: ADPRT3, ADPRTL3, PARP3
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4l6za1, d4l6za2, d4l6za3 - Heterogens: 1DC, DMS, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4l6zA (A:)
smkrvqpcsldpatqklitnifskemfkntmalmdldvkkmplgklskqqiargfealea
leealkgptdggqsleelsshfytviphnfghsqpppinspellqakkdmllvladiela
qalqavseqektveevphpldrdyqllkcqlqlldsgapeykviqtyleqtgsnhrcptl
qhiwkvnqegeedrfqahsklgnrkllwhgtnmavvaailtsglrimphsggrvgkgiyf
asensksagyvigmkcgahhvgymflgevalgrehhintdnpslkspppgfdsviarght
epdptqdteleldgqqvvvpqgqpvpcpefssstfsqseyliyqesqcrlryllevh
Sequence, based on observed residues (ATOM records): (download)
>4l6zA (A:)
smkrvqpcsldpatqklitnifskemfkntmalmdldvkkmplgklskqqiargfealea
leealkdggqsleelsshfytviphnfghsqpppinspellqakkdmllvladielaqal
qavseqektveevphpldrdyqllkcqlqlldsgapeykviqtyleqtgsnhrcptlqhi
wkvnqegeedrfqahsklgnrkllwhgtnmavvaailtsglrimphsggrvgkgiyfase
nsksagyvigmkcgahhvgymflgevalgrehhintdnpslkspppgfdsviarghtepd
ptqdteleldgqqvvvpqgqpvpcpefssstfsqseyliyqesqcrlryllevh