PDB entry 4l5b
View 4l5b on RCSB PDB site
Description: Human dCK C4S-S74E mutant in complex with UDP and the DI-43 inhibitor
Class: transferase/transferase inhibitor
Keywords: phosphoryl transfer, phosphorylation, deoxycytidine kinase, transferase-transferase inhibitor complex
Deposited on
2013-06-10, released
2013-09-18
The last revision prior to the SCOPe 2.08 freeze date was dated
2013-11-27, with a file datestamp of
2013-11-22.
Experiment type: XRAY
Resolution: 1.94 Å
R-factor: 0.19
AEROSPACI score: 0.37
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Deoxycytidine kinase
Species: Homo sapiens [TaxId:9606]
Gene: DCK
Database cross-references and differences (RAF-indexed):
- Uniprot P27707 (Start-279)
- engineered mutation (64)
- engineered mutation (78)
- engineered mutation (93)
- engineered mutation (165)
Domains in SCOPe 2.08: d4l5ba_ - Chain 'B':
Compound: Deoxycytidine kinase
Species: Homo sapiens [TaxId:9606]
Gene: DCK
Database cross-references and differences (RAF-indexed):
- Uniprot P27707 (Start-279)
- engineered mutation (64)
- engineered mutation (78)
- engineered mutation (93)
- engineered mutation (165)
Domains in SCOPe 2.08: d4l5bb_ - Heterogens: 1UX, UDP, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4l5bA (A:)
mgsshhhhhhssglvprgshmatppkrsspsfsassegtrikkisiegniaagkstfvni
lkqlsedwevvpepvarwsnvqstqdefeeltmeqknggnvlqmmyekperwsftfqtya
clsriraqlaslngklkdaekpvlffersvysdryifasnlyesesmnetewtiyqdwhd
wmnnqfgqsleldgiiylqatpetclhriylrgrneeqgipleyleklhykheswllhrt
lktnfdylqevpiltldvnedfkdkyeslvekvkeflstl
Sequence, based on observed residues (ATOM records): (download)
>4l5bA (A:)
rikkisiegniaagkstfvnilkqlsedwevvpepvarwsnltmeqknggnvlqmmyekp
erwsftfqtyaclsriraqlaslngklkdaekpvlffersvysdryifasnlyesesmne
tewtiyqdwhdwmnnqfgqsleldgiiylqatpetclhriylrgrneeqgipleyleklh
ykheswllhrtlktnfdylqevpiltldvnedfkdkyeslvekvkeflstl
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4l5bB (B:)
mgsshhhhhhssglvprgshmatppkrsspsfsassegtrikkisiegniaagkstfvni
lkqlsedwevvpepvarwsnvqstqdefeeltmeqknggnvlqmmyekperwsftfqtya
clsriraqlaslngklkdaekpvlffersvysdryifasnlyesesmnetewtiyqdwhd
wmnnqfgqsleldgiiylqatpetclhriylrgrneeqgipleyleklhykheswllhrt
lktnfdylqevpiltldvnedfkdkyeslvekvkeflstl
Sequence, based on observed residues (ATOM records): (download)
>4l5bB (B:)
rikkisiegniaagkstfvnilkqlsedwevvpepvarwsltmeqknggnvlqmmyekpe
rwsftfqtyaclsriraqlaslngklkdaekpvlffersvysdryifasnlyesesmnet
ewtiyqdwhdwmnnqfgqsleldgiiylqatpetclhriylrgrneeqgipleyleklhy
kheswllhrtlktnfdylqevpiltldvnedfkdkyeslvekvkeflstl