PDB entry 4jt3

View 4jt3 on RCSB PDB site
Description: Crystal Structure of TTK kinase domain with an inhibitor: 400740
Class: Transferase/Transferase Inhibitor
Keywords: Transferase-Transferase Inhibitor complex
Deposited on 2013-03-22, released 2014-03-26
The last revision prior to the SCOPe 2.03 freeze date was dated 2014-03-26, with a file datestamp of 2014-03-21.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: 0.239
AEROSPACI score: 0.27 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Dual specificity protein kinase TTK
    Species: Homo sapiens [TaxId:9606]
    Gene: TTK, MPS1, MPS1L1
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.03: d4jt3a_
  • Heterogens: PO4, 1PH, EDO, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >4jt3A (A:)
    necisvkgriysilkqigsggsskvfqvlnekkqiyaikyvnleeadnqtldsyrneiay
    lnklqqhsdkiirlydyeitdqyiymvmecgnidlnswlkkkksidpwerksywknmlea
    vhtihqhgivhsdlkpanflivdgmlklidfgianqmqpdttsvvkdsqvgtvnymppea
    ikdmsssrengkskskispksdvwslgcilyymtygktpfqqiinqisklhaiidpnhei
    efpdipekdlqdvlkcclkrdpkqrisipellahpyvqiqt
    

    Sequence, based on observed residues (ATOM records): (download)
    >4jt3A (A:)
    necisvkgriysilkqigsggsskvfqvlnekkqiyaikyvnleeadnqtldsyrneiay
    lnklqqhsdkiirlydyeitdqyiymvmecgnidlnswlkkkksidpwerksywknmlea
    vhtihqhgivhsdlkpanflivdgmlklidfgianqmgtvnymppeaikdmspksdvwsl
    gcilyymtygktpfqqiinqisklhaiidpnheiefpdipekdlqdvlkcclkrdpkqri
    sipellahpyvqiq