PDB entry 4i41
View 4i41 on RCSB PDB site
Description: Crystal Structure of human Ser/Thr kinase Pim1 in complex with mitoxantrone
Class: transferase/transferase inhibitor
Keywords: Ser/Thr kinase, mitoxantrone, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2012-11-27, released
2013-12-11
The last revision prior to the SCOPe 2.05 freeze date was dated
2013-12-11, with a file datestamp of
2013-12-06.
Experiment type: XRAY
Resolution: 2.7 Å
R-factor: 0.2
AEROSPACI score: 0.22
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase pim-1
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d4i41a_ - Heterogens: MIX, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4i41A (A:)
gphmkekeplesqyqvgpllgsggfgsvysgirvsdnlpvaikhvekdrisdwgelpngt
rvpmevvllkkvssgfsgvirlldwferpdsfvlilerpepvqdlfdfitergalqeela
rsffwqvleavrhchncgvlhrdikdenilidlnrgelklidfgsgallkdtvytdfdgt
rvysppewiryhryhgrsaavwslgillydmvcgdipfehdeeiirgqvffrqrvssecq
hlirwclalrpsdrptfeeiqnhpwmqdvllpqetaeihlh
Sequence, based on observed residues (ATOM records): (download)
>4i41A (A:)
plesqyqvgpllgsggfgsvysgirvsdnlpvaikhvekdrisdwgelpngtrvpmevvl
lkkvssgfsgvirlldwferpdsfvlilerpepvqdlfdfitergalqeelarsffwqvl
eavrhchncgvlhrdikdenilidlnrgelklidfgsgallkdtvytdfdgtrvysppew
iryhryhgrsaavwslgillydmvcgdipfehdeeiirgqvffrqrvssecqhlirwcla
lrpsdrptfeeiqnhpwmqdvllpqetaeihlh