PDB entry 4i23
View 4i23 on RCSB PDB site
Description: Crystal structure of the wild-type EGFR kinase domain in complex with dacomitinib (soaked)
Class: transferase
Keywords: Kinase domain, Phosphotransfer, ATP binding, TRANSFERASE
Deposited on
2012-11-21, released
2013-01-16
The last revision prior to the SCOPe 2.02 freeze date was dated
2013-02-27, with a file datestamp of
2013-02-22.
Experiment type: XRAY
Resolution: 2.8 Å
R-factor: 0.229
AEROSPACI score: 0.25
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Epidermal growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: EGFR, ERBB, ERBB1, HER1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d4i23a_ - Heterogens: 1C9
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4i23A (A:)
gsgeapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelreatsp
kankeildeayvmasvdnphvcrllgicltstvqlitqlmpfgclldyvrehkdnigsqy
llnwcvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfglakllgaeekeyhaeg
gkvpikwmalesilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekgerl
pqppictidvymimvkcwmidadsrpkfreliiefskmardpqrylviqgdermhlpspt
dsnfyralmdeedmddvvdadeylipqqg
Sequence, based on observed residues (ATOM records): (download)
>4i23A (A:)
sgeapnqallrilketefkkikvlgsgtvykglwipegekvkipvaikelatspkankei
ldeayvmasvdnphvcrllgicltstvqlitqlmpfgclldyvrehkdnigsqyllnwcv
qiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfglakllgaeekeyhaeggkvpik
wmalesilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekgerlpqppic
tidvymimvkcwmidadsrpkfreliiefskmardpqrylviqgdermhlpdmddvvdad
eyli