PDB entry 4hxs
View 4hxs on RCSB PDB site
Description: Brd4 Bromodomain 1 complex with N-[3-(2-OXO-2,3-DIHYDRO-1,3-THIAZOL-4-YL)PHENYL]-1-PHENYLMETHANESULFONAMIDE inhibitor
Class: protein binding/inhibitor
Keywords: BRD4, Bromodomain, four alpha helices, PROTEIN BINDING-INHIBITOR complex
Deposited on
2012-11-12, released
2013-04-03
The last revision prior to the SCOPe 2.03 freeze date was dated
2013-06-19, with a file datestamp of
2013-06-14.
Experiment type: XRAY
Resolution: 1.43 Å
R-factor: 0.179
AEROSPACI score: 0.68
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Bromodomain-containing protein 4
Species: Homo sapiens [TaxId:9606]
Gene: BRD4, HUNK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d4hxsa_ - Heterogens: 1A3, HOH