PDB entry 4gv2
View 4gv2 on RCSB PDB site
Description: Human ARTD3 (PARP3) - Catalytic domain in complex with inhibitor ME0354
Class: transferase/transferase inhibitor
Keywords: nad, ADP-ribose, parp3, artd3, artd transferase domain, ADP- ribosylation, transferase-transferase inhibitor complex, transferase, ADP-ribosylation
Deposited on
2012-08-30, released
2013-06-19
The last revision prior to the SCOPe 2.05 freeze date was dated
2013-10-16, with a file datestamp of
2013-10-11.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: 0.163
AEROSPACI score: 0.54
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Poly [ADP-ribose] polymerase 3
Species: Homo sapiens [TaxId:9606]
Gene: PARP3
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d4gv2a1, d4gv2a2 - Heterogens: 5ME, DMS, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4gv2A (A:)
smkrvqpcsldpatqklitnifskemfkntmalmdldvkkmplgklskqqiargfealea
leealkgptdggqsleelsshfytviphnfghsqpppinspellqakkdmllvladiela
qalqavseqektveevphpldrdyqllkcqlqlldsgapeykviqtyleqtgsnhrcptl
qhiwkvnqegeedrfqahsklgnrkllwhgtnmavvaailtsglrimphsggrvgkgiyf
asensksagyvigmkcgahhvgymflgevalgrehhintdnpslkspppgfdsviarght
epdptqdteleldgqqvvvpqgqpvpcpefssstfsqseyliyqesqcrlryllevh
Sequence, based on observed residues (ATOM records): (download)
>4gv2A (A:)
smkrvqpcsldpatqklitnifskemfkntmalmdldvkkmplgklskqqiargfealea
leealkdggqsleelsshfytviphnfghsqpppinspellqakkdmllvladielaqal
qavseqektveevphpldrdyqllkcqlqlldsgapeykviqtyleqtgsnhrcptlqhi
wkvnqegeedrfqahsklgnrkllwhgtnmavvaailtsglrimphsggrvgkgiyfase
nsksagyvigmkcgahhvgymflgevalgrehhintdnpslkspppgfdsviarghtepd
ptqdteleldgqqvvvpqgqpvpcpefssstfsqseyliyqesqcrlryllevh