PDB entry 4g2i
View 4g2i on RCSB PDB site
Description: Structural basis for the accommodation of bis- and tris-aromatic derivatives in Vitamin D Nuclear Receptor
Class: transcription/transcription inhibitor
Keywords: VDR, transcription regulation, nuclear receptor, alpha helical sandwich, ligand, DNA, phosphorylation, nucleus, transcription-transcription inhibitor complex
Deposited on
2012-07-12, released
2012-09-26
The last revision prior to the SCOPe 2.08 freeze date was dated
2012-11-21, with a file datestamp of
2012-11-16.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: 0.195
AEROSPACI score: 0.53
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Vitamin D3 receptor
Species: Homo sapiens [TaxId:9606]
Gene: Vdr, Nr1i1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4g2ia_ - Heterogens: 0VQ, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4g2iA (A:)
dslrpklseeqqriiailldahhktydptysdfcqfrppvrvndgggsvtlelsqlsmlp
hladlvsysiqkvigfakmipgfrdltsedqivllkssaievimlrsnesftmddmswtc
gnqdykyrvsdvtkaghslelieplikfqvglkklnlheeehvllmaicivspdrpgvqd
aalieaiqdrlsntlqtyircrhpppgshllyakmiqkladlrslneehskqyrclsfqp
ecsmkltplvlevfgneis
Sequence, based on observed residues (ATOM records): (download)
>4g2iA (A:)
lrpklseeqqriiailldahhktydptysdfcqfrppvrvndgggsvtlelsqlsmlphl
adlvsysiqkvigfakmipgfrdltsedqivllkssaievimlrsnesftmddmswtcgn
qdykyrvsdvtkaghslelieplikfqvglkklnlheeehvllmaicivspdrpgvqdaa
lieaiqdrlsntlqtyircrhpppgshllyakmiqkladlrslneehskqyrclsfqpec
smkltplvlevfg