PDB entry 4g17
View 4g17 on RCSB PDB site
Description: Crystal structure of ck1g3 with 2-[(4-TERT-BUTYLPHENYL)AMINO]-1H-BENZIMIDAZOLE-6-CARBONITRILE
Class: TRANSFERASE/TRANSFERASE inhibitor
Keywords: ck1g, kinase, inhibitor, TRANSFERASE-TRANSFERASE inhibitor complex
Deposited on
2012-07-10, released
2013-05-22
The last revision prior to the SCOPe 2.04 freeze date was dated
2013-05-22, with a file datestamp of
2013-05-17.
Experiment type: XRAY
Resolution: 2.1 Å
R-factor: 0.219
AEROSPACI score: 0.39
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: casein kinase I isoform gamma-3
Species: Homo sapiens [TaxId:9606]
Gene: CSNK1G3
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.04: d4g17a_ - Heterogens: 0VN, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4g17A (A:)
gsgvlmvgpnfrvgkkigcgnfgelrlgknlytneyvaiklepmksrapqlhleyrfykq
lgsgdgipqvyyfgpcgkynamvlellgpsledlfdlcdrtfslktvlmiaiqlisrmey
vhsknliyrdvkpenfligrpgnktqqvihiidfglakeyidpetkkhipyrehksltgt
arymsinthlgkeqsrrddlealghmfmyflrgslpwqglkadtlkeryqkigdtkratp
ievlcenfpematylryvrrldffekpdydylrklftdlfdrkgymfdyeydwigkqlpt
pvgavqqdpalssnreahqhrdkmqqsknq
Sequence, based on observed residues (ATOM records): (download)
>4g17A (A:)
gsgvlmvgpnfrvgkkigcgnfgelrlgknlytneyvaiklepmksrapqlhleyrfykq
lgsgdgipqvyyfgpcgkynamvlellgpsledlfdlcdrtfslktvlmiaiqlisrmey
vhsknliyrdvkpenfligrpgnktqqvihiidfglakeyidpetkkhipyrehksltgt
arymsinthlgkeqsrrddlealghmfmyflrgslpwqglkadtlkeryqkigdtkratp
ievlcenfpematylryvrrldffekpdydylrklftdlfdrkgymfdyeydwigkqlpt
pv