PDB entry 4ft3
View 4ft3 on RCSB PDB site
Description: Crystal Structure of the CHK1
Class: TRANSFERASE/TRANSFERASE inhibitor
Keywords: TRANSFERASE, TRANSFERASE-TRANSFERASE inhibitor complex
Deposited on
2012-06-27, released
2012-08-22
The last revision prior to the SCOPe 2.03 freeze date was dated
2012-08-22, with a file datestamp of
2012-08-17.
Experiment type: XRAY
Resolution: 2.5 Å
R-factor: 0.17
AEROSPACI score: 0.37
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase Chk1
Species: Homo sapiens [TaxId:9606]
Gene: CHEK1, CHK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d4ft3a_ - Heterogens: H1K, SO4, GOL, IPA, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4ft3A (A:)
avpfvedwdlvqtlgegaygevqlavnrvteeavavkivdmkravdcpenikkeicinkm
lnhenvvkfyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvyl
hgigithrdikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkr
refhaepvdvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplal
lhkilvenpsaritipdikkdrwynkplkkgakrprvts
Sequence, based on observed residues (ATOM records): (download)
>4ft3A (A:)
avpfvedwdlvqtlgegaygevqlavnrvteeavavkivdmenikkeicinkmlnhenvv
kfyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvylhgigith
rdikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkrrefhaep
vdvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplallhkilve
npsaritipdikkdrwynkplkkgakrprvts