PDB entry 4fsn

View 4fsn on RCSB PDB site
Description: Crystal Structure of the CHK1
Class: TRANSFERASE/TRANSFERASE inhibitor
Keywords: TRANSFERASE, TRANSFERASE-TRANSFERASE inhibitor complex
Deposited on 2012-06-27, released 2012-08-22
The last revision prior to the SCOPe 2.06 freeze date was dated 2013-05-29, with a file datestamp of 2013-05-24.
Experiment type: XRAY
Resolution: 2.1 Å
R-factor: 0.178
AEROSPACI score: 0.44 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Serine/threonine-protein kinase Chk1
    Species: Homo sapiens [TaxId:9606]
    Gene: CHEK1, CHK1
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.06: d4fsna_
  • Heterogens: A58, SO4, IPA, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >4fsnA (A:)
    apfvedwdlvqtlgegaygevqlavnrvteeavavkivdmkravdcpenikkeicinkml
    nhenvvkfyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvylh
    gigithrdikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkrr
    efhaepvdvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplall
    hkilvenpsaritipdikkdrwynkplkkgakrprvts
    

    Sequence, based on observed residues (ATOM records): (download)
    >4fsnA (A:)
    apfvedwdlvqtlgegagevqlavnrvteeavavkivdmenikkeicinkmlnhenvvkf
    yghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvylhgigithrd
    ikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkrrefhaepvd
    vwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplallhkilvenp
    saritipdikkdrwynkplkkgakrprvts