PDB entry 4ewh
View 4ewh on RCSB PDB site
Description: Co-crystal structure of ACK1 with inhibitor
Class: transferase/transferase inhibitor
Keywords: Drug Design, Enzyme Inhibitors, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2012-04-27, released
2012-09-19
The last revision prior to the SCOPe 2.02 freeze date was dated
2012-10-31, with a file datestamp of
2012-10-26.
Experiment type: XRAY
Resolution: 2.5 Å
R-factor: 0.259
AEROSPACI score: 0.24
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Activated CDC42 kinase 1
Species: Homo sapiens [TaxId:9606]
Gene: TNK2, ACK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d4ewha_ - Chain 'B':
Compound: Activated CDC42 kinase 1
Species: Homo sapiens [TaxId:9606]
Gene: TNK2, ACK1
Database cross-references and differences (RAF-indexed):
- Heterogens: T77, HOH