PDB entry 4eev
View 4eev on RCSB PDB site
Description: Crystal structure of c-Met in complex with LY2801653
Class: transferase/transferase inhibitor
Keywords: protein tyrosine kinase, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2012-03-28, released
2013-04-10
The last revision prior to the SCOPe 2.03 freeze date was dated
2013-09-04, with a file datestamp of
2013-08-30.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: 0.19
AEROSPACI score: 0.52
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Hepatocyte growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: MET
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d4eeva_ - Heterogens: L1X, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4eevA (A:)
mhhhhhhmgdsdisspllqntvhidlsalnpelvqavqhvvigpsslivhfnevigrghf
gcvyhgtlldndgkkihcavkslnritdigevsqfltegiimkdfshpnvlsllgiclrs
egsplvvlpymkhgdlrnfirnethnptvkdligfglqvakgmkylaskkfvhrdlaarn
cmldekftvkvadfglardmydkeyysvhnktgaklpvkwmaleslqtqkfttksdvwsf
gvllwelmtrgappypdvntfditvyllqgrrllqpeycpdplyevmlkcwhpkaemrps
fselvsrisaifstfig
Sequence, based on observed residues (ATOM records): (download)
>4eevA (A:)
pllqntvhidlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlldndgkk
ihcavkslnritdigevsqfltegiimkdfshpnvlsllgiclrsegsplvvlpymkhgd
lrnfirnethnptvkdligfglqvakgmkylaskkfvhrdlaarncmldekftvkvadfg
klpvkwmaleslqtqkfttksdvwsfgvllwelmtrgappypdvntfditvyllqgrrll
qpeycpdplyevmlkcwhpkaemrpsfselvsrisaifstfig