PDB entry 4e20
View 4e20 on RCSB PDB site
Description: Structure of mouse Tyk-2 complexed to a 3-aminoindazole inhibitor
Class: transferase/transferase inhibitor
Keywords: kinase catalytic domain, kinase, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2012-03-07, released
2012-10-03
The last revision prior to the SCOPe 2.05 freeze date was dated
2012-10-03, with a file datestamp of
2012-09-28.
Experiment type: XRAY
Resolution: 2.6 Å
R-factor: 0.2
AEROSPACI score: 0.31
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Non-receptor tyrosine-protein kinase TYK2
Species: Mus musculus [TaxId:10090]
Gene: TYK2
Database cross-references and differences (RAF-indexed):
- Uniprot Q9R117 (0-289)
- engineered mutation (135)
Domains in SCOPe 2.05: d4e20a_ - Heterogens: 0MY, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4e20A (A:)
dptvfhkrylkkirdlgeghfgkvslycydptndgtgemvavkalkegcgpqlrsgwqre
ieilrtlyhehivkykgccedqgeksvqlvmeyvplgslrdylprhcvglaqlllfaqqi
cegmaylhaqhyihralaarnvlldndrlvkigdfglakavpegheyyrvredgdspvfw
yapeclkeckfyyasdvwsfgvtlyelltycdsnqsphtkftelightqgqmtvlrltel
lergerlprpdrcpceiyhlmkncweteasfrptfqnlvpilqtaqekyq
Sequence, based on observed residues (ATOM records): (download)
>4e20A (A:)
dptvfhkrylkkirdlgeghfgkvslycydptndgtgemvavkalkegcgpqlrsgwqre
ieilrtlyhehivkykgccedsvqlvmeyvplgslrdylprhcvglaqlllfaqqicegm
aylhaqhyihralaarnvlldndrlvkigdfglakavpegheyyrvredgdspvfwyape
clkeckfyyasdvwsfgvtlyelltycdsnqsphtkfteligqmtvlrltellergerlp
rpdrcpceiyhlmkncweteasfrptfqnlvpilqtaqekyq