PDB entry 4dhf
View 4dhf on RCSB PDB site
Description: Structure of Aurora A mutant bound to Biogenidec cpd 15
Class: transferase/transferase inhibitor
Keywords: Ser/Thr kinase mitotic kinase pyrazolopyrimidine, phosphorylation, TPX2, transferase-transferase inhibitor complex
Deposited on
2012-01-27, released
2012-07-18
The last revision prior to the SCOPe 2.06 freeze date was dated
2012-07-18, with a file datestamp of
2012-07-13.
Experiment type: XRAY
Resolution: 2.8 Å
R-factor: 0.21
AEROSPACI score: 0.24
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Aurora kinase A
Species: Homo sapiens [TaxId:9606]
Gene: AIK, AIRK1, ARK1, AURA, AURKA, AuroraA, AYK1, BTAK, IAK1, STK15, STK6
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d4dhfa_ - Chain 'B':
Compound: Aurora kinase A
Species: Homo sapiens [TaxId:9606]
Gene: AIK, AIRK1, ARK1, AURA, AURKA, AuroraA, AYK1, BTAK, IAK1, STK15, STK6
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d4dhfb_ - Heterogens: 0K6, PO4, MG
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4dhfA (A:)
gplgsrqwaledfeigrplgkgkfgnvylarekqskfilalkvlfkaqlekagvehqlrr
eveiqshlrhpnilrlygyfhdatrvylileyaplgtvyrelqklskfdeqrtatyitel
analsychskrvihrdikpenlllgsagelkiadfgwsvhapssrrddlcgtldylppem
iegrmhdekvdlwslgvlcyeflvgkppfeantyqetykrisrveftfpdfvtegardli
srllkhnpsqrpmlrevlehpwitansskps
Sequence, based on observed residues (ATOM records): (download)
>4dhfA (A:)
waledfeigrplgkgkfgnvylarekqskfilalkvlfkaqlekagvehqlrreveiqsh
lrhpnilrlygyfhdatrvylileyaplgtvyrelqklskfdeqrtatyitelanalsyc
hskrvihrdikpenlllgsagelkiadfgwsvhapssrcgtldylppemiegrmhdekvd
lwslgvlcyeflvgkppfeantyqetykrisrveftfpdfvtegardlisrllkhnpsqr
pmlrevlehpwitanssk
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4dhfB (B:)
gplgsrqwaledfeigrplgkgkfgnvylarekqskfilalkvlfkaqlekagvehqlrr
eveiqshlrhpnilrlygyfhdatrvylileyaplgtvyrelqklskfdeqrtatyitel
analsychskrvihrdikpenlllgsagelkiadfgwsvhapssrrddlcgtldylppem
iegrmhdekvdlwslgvlcyeflvgkppfeantyqetykrisrveftfpdfvtegardli
srllkhnpsqrpmlrevlehpwitansskps
Sequence, based on observed residues (ATOM records): (download)
>4dhfB (B:)
waledfeigrplgkgkfgnvylarekqskfilalkvlfkaqlekagvehqlrreveiqsh
lrhpnilrlygyfhdatrvylileyaplgtvyrelqklskfdeqrtatyitelanalsyc
hskrvihrdikpenlllgsagelkiadfgwsvhapssrcgtldylppemiegrmhdekvd
lwslgvlcyeflvgkppfeantyqetykrisrveftfpdfvtegardlisrllkhnpsqr
pmlrevlehpwitanssk