PDB entry 4dbn
View 4dbn on RCSB PDB site
Description: Crystal Structure of the Kinase domain of Human B-raf with a [1,3]thiazolo[5,4-b]pyridine derivative
Class: transferase/transferase inhibitor
Keywords: kinase drug complex, Ser/Thr Kinase, ATP Binding, Phosphorylation, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2012-01-16, released
2012-04-11
The last revision prior to the SCOPe 2.05 freeze date was dated
2012-06-13, with a file datestamp of
2012-06-08.
Experiment type: XRAY
Resolution: 3.15 Å
R-factor: 0.198
AEROSPACI score: 0.24
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase B-raf
Species: Homo sapiens [TaxId:9606]
Gene: BRAF, BRAF1, P94, RAFB1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d4dbna_ - Chain 'B':
Compound: Serine/threonine-protein kinase B-raf
Species: Homo sapiens [TaxId:9606]
Gene: BRAF, BRAF1, P94, RAFB1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d4dbnb_ - Heterogens: 0JA, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4dbnA (A:)
gsdssddweipdgqitvgqrigsgsfgtvykgkwhgdvavkmlnvtaptpqqlqafknev
gvlrktrhvnillfmgystkpqlaivtqwcegsslyhhlhiietkfemiklidiarqtaq
gmdylhaksiihrdlksnniflhedltvkigdfglatvksrwsgshqfeqlsgsilwmap
evirmqdknpysfqsdvyafgivlyelmtgqlpysninnrdqiifmvgrgylspdlskvr
sncpkamkrlmaeclkkkrderplfpqilasiellarslpkihr
Sequence, based on observed residues (ATOM records): (download)
>4dbnA (A:)
ddweipdgqitvgqrigsgsfgtvykgkwhgdvavkmlnvtaptpqqlqafknevgvlrk
trhvnillfmgystkpqlaivtqwcegsslyhhlhiietkfemiklidiarqtaqgmdyl
haksiihrdlksnniflhedltvkigdfglgsilwmapevirmqdknpysfqsdvyafgi
vlyelmtgqlpysninnrdqiifmvgrgylspdlskvrsncpkamkrlmaeclkkkrder
plfpqilasiellarsl
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4dbnB (B:)
gsdssddweipdgqitvgqrigsgsfgtvykgkwhgdvavkmlnvtaptpqqlqafknev
gvlrktrhvnillfmgystkpqlaivtqwcegsslyhhlhiietkfemiklidiarqtaq
gmdylhaksiihrdlksnniflhedltvkigdfglatvksrwsgshqfeqlsgsilwmap
evirmqdknpysfqsdvyafgivlyelmtgqlpysninnrdqiifmvgrgylspdlskvr
sncpkamkrlmaeclkkkrderplfpqilasiellarslpkihr
Sequence, based on observed residues (ATOM records): (download)
>4dbnB (B:)
ddweipdgqitvgqrigsgsfgtvykgkwhgdvavkmlnvtaptpqqlqafknevgvlrk
trhvnillfmgystkpqlaivtqwcegsslyhhlhiietkfemiklidiarqtaqgmdyl
haksiihrdlksnniflhedltvkigdfglatvksrwgsilwmapevirmqdknpysfqs
dvyafgivlyelmtgqlpysninnrdqiifmvgrgylspdlskvrsncpkamkrlmaecl
kkkrderplfpqilasiellars