PDB entry 4cmo
View 4cmo on RCSB PDB site
Description: Structure of the Human Anaplastic Lymphoma Kinase in Complex with the inhibitor 2-((1R)-1-((3-amino-6-(2-methoxypyridin-3-yl)pyrazin-2-yl) oxy)ethyl)-4-fluoro-N-methylbenzamide
Class: transferase
Keywords: transferase, receptor tyrosine kinase inhibitor
Deposited on
2014-01-16, released
2014-05-28
The last revision prior to the SCOPe 2.05 freeze date was dated
2014-06-25, with a file datestamp of
2014-06-20.
Experiment type: XRAY
Resolution: 1.83 Å
R-factor: 0.199
AEROSPACI score: 0.41
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: ALK tyrosine kinase receptor
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d4cmoa_ - Heterogens: YPW, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4cmoA (A:)
mahhhhhhnpnycfagktssisdlkevprknitlirglghgafgevyegqvsgmpndpsp
lqvavktlpevcseqdeldflmealiiskfnhqnivrcigvslqslprfillelmaggdl
ksflretrprpsqpsslamldllhvardiacgcqyleenhfihrdiaarnclltcpgpgr
vakigdfgmardiyrasyyrkggcamlpvkwmppeafmegiftsktdtwsfgvllweifs
lgympypsksnqevlefvtsggrmdppkncpgpvyrimtqcwqhqpedrpnfaiilerie
yctqdpdvintalpieygplveeeekv
Sequence, based on observed residues (ATOM records): (download)
>4cmoA (A:)
npnycfagktssisdlkevprknitlirglghgafgevyegqvplqvavktlpevcseqd
eldflmealiiskfnhqnivrcigvslqslprfillelmaggdlksflretrprpsqpss
lamldllhvardiacgcqyleenhfihrdiaarnclltcpgpgrvakigdfgmardiyrg
gcamlpvkwmppeafmegiftsktdtwsfgvllweifslgympypsksnqevlefvtsgg
rmdppkncpgpvyrimtqcwqhqpedrpnfaiilerieyctqdpdvintalpieyg