PDB entry 4bzn
View 4bzn on RCSB PDB site
Description: Crystal structure of PIM1 in complex with a Pyrrolo(1,2-a)Pyrazinone inhibitor
Class: transferase
Keywords: pim1, ATP binding, kinase inhibitor, transferase
Deposited on
2013-07-29, released
2013-10-30
The last revision prior to the SCOPe 2.04 freeze date was dated
2013-11-13, with a file datestamp of
2013-11-08.
Experiment type: XRAY
Resolution: 1.9 Å
R-factor: 0.17766
AEROSPACI score: 0.42
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase pim-1
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.04: d4bzna_ - Heterogens: UGX, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4bznA (A:)
gpllskinslahlraapcndlhatklapgkekeplesqyqvgpllgsggfgsvysgirvs
dnlpvaikhvekdrisdwgelpngtrvpmevvllkkvssgfsgvirlldwferpdsfvli
lerpepvqdlfdfitergalqeelarsffwqvleavrhchncgvlhrdikdenilidlnr
gelklidfgsgallkdtvytdfdgtrvysppewiryhryhgrsaavwslgillydmvcgd
ipfehdeeiirgqvffrqrvssecqhlirwclalrpsdrptfeeiqnhpwmqdvllpqet
aeihlhslspgpsk
Sequence, based on observed residues (ATOM records): (download)
>4bznA (A:)
plesqyqvgpllgsggfgsvysgirvsdnlpvaikhvekdrisdwgelpngtrvpmevvl
lkkvssgfsgvirlldwferpdsfvlilerpepvqdlfdfitergalqeelarsffwqvl
eavrhchncgvlhrdikdenilidlnrgelklidfgsgallkdtvytdfdgtrvysppew
iryhryhgrsaavwslgillydmvcgdipfehdeeiirgqvffrqrvssecqhlirwcla
lrpsdrptfeeiqnhpwmqdvllpqetaeihlh