PDB entry 4btt
View 4btt on RCSB PDB site
Description: factor Xa in complex with the dual thrombin-FXa inhibitor 31.
Class: hydrolase
Keywords: hydrolase, sar107375, factor xa inhibitor, thrombin inhibitor, chlorothiophene p1 fragment, s3 subsite, microsomes stability, oral antithrombotic, dual inhibitor, IV antithrombotic
Deposited on
2013-06-19, released
2013-12-18
The last revision prior to the SCOPe 2.07 freeze date was dated
2014-01-15, with a file datestamp of
2014-01-10.
Experiment type: XRAY
Resolution: 2.59 Å
R-factor: 0.201
AEROSPACI score: 0.24
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: coagulation factor x light chain
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4btta_ - Chain 'B':
Compound: coagulation factor x
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4bttb_ - Chain 'E':
Compound: coagulation factor x light chain
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4btte_ - Chain 'F':
Compound: coagulation factor x
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4bttf_ - Heterogens: CA, VYR, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4bttA (A:)
ykdgdqcetspcqnqgkckdglgeytctclegfegkncelftrklcsldngdcdqfchee
qnsvvcscargytladngkaciptgpypcgkqtler
Sequence, based on observed residues (ATOM records): (download)
>4bttA (A:)
rklcsldngdcdqfcheeqnsvvcscargytladngkaciptgpypcgkqt
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4bttB (B:)
ivggqeckdgecpwqallineenegfcggtilsefyiltaahclyqakrfkvrvgdrnte
qeeggeavhevevvikhnrftketydfdiavlrlktpitfrmnvapaclperdwaestlm
tqktgivsgfgrthekgrqstrlkmlevpyvdrnscklsssfiitqnmfcagydtkqeda
cqgdsggphvtrfkdtyfvtgivswgegcarkgkygiytkvtaflkwidrsmktrglpka
kshapevitssplk
Sequence, based on observed residues (ATOM records): (download)
>4bttB (B:)
ivggqeckdgecpwqallineenegfcggtilsefyiltaahclyqakrfkvrvgdrnte
qeeggeavhevevvikhnrftketydfdiavlrlktpitfrmnvapaclperdwaestlm
tqktgivsgfgrthekgrqstrlkmlevpyvdrnscklsssfiitqnmfcagydtkqeda
cqgdsggphvtrfkdtyfvtgivswgegcarkgkygiytkvtaflkwidrsmktr
- Chain 'E':
Sequence, based on SEQRES records: (download)
>4bttE (E:)
ykdgdqcetspcqnqgkckdglgeytctclegfegkncelftrklcsldngdcdqfchee
qnsvvcscargytladngkaciptgpypcgkqtler
Sequence, based on observed residues (ATOM records): (download)
>4bttE (E:)
klcsldngdcdqfcheeqnsvvcscargytladngkaciptgpypcgkqtler
- Chain 'F':
Sequence, based on SEQRES records: (download)
>4bttF (F:)
ivggqeckdgecpwqallineenegfcggtilsefyiltaahclyqakrfkvrvgdrnte
qeeggeavhevevvikhnrftketydfdiavlrlktpitfrmnvapaclperdwaestlm
tqktgivsgfgrthekgrqstrlkmlevpyvdrnscklsssfiitqnmfcagydtkqeda
cqgdsggphvtrfkdtyfvtgivswgegcarkgkygiytkvtaflkwidrsmktrglpka
kshapevitssplk
Sequence, based on observed residues (ATOM records): (download)
>4bttF (F:)
ivggqeckdgecpwqallineenegfcggtilsefyiltaahclyqakrfkvrvgdrnte
qeeggeavhevevvikhnrftketydfdiavlrlktpitfrmnvapaclperdwaestlm
tqktgivsgfgrthekgrqstrlkmlevpyvdrnscklsssfiitqnmfcagydtkqeda
cqgdsggphvtrfkdtyfvtgivswgegcarkgkygiytkvtaflkwidrsmktr