PDB entry 4bky
View 4bky on RCSB PDB site
Description: Crystal structure of unphosphorylated Maternal Embryonic Leucine zipper Kinase (MELK) in complex with pyrrolopyrazole inhibitor
Class: transferase
Keywords: transferase
Deposited on
2013-04-30, released
2013-08-21
The last revision prior to the SCOPe 2.07 freeze date was dated
2019-04-24, with a file datestamp of
2019-04-19.
Experiment type: XRAY
Resolution: 1.83 Å
R-factor: 0.20392
AEROSPACI score: 0.49
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: maternal embryonic leucine zipper kinase
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4bkya_ - Heterogens: 82B, UNX, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4bkyA (A:)
gpkdydellkyyelhetigtggfakvklachiltgemvaikimdkntlgsdlprikteie
alknlrhqhicqlyhvletankifmvleycpggelfdyiisqdrlseeetrvvfrqivsa
vayvhsqgyahrdlkpenllfdeyhklklidfglcakpkgnkdyhlqtccgslayaapel
iqgksylgseadvwsmgillyvlmcgflpfdddnvmalykkimrgkydvpkwlspssill
lqqmlqvdpkkrismknllnhpwimqdynypvewqsknpfihldddcvtelsvhhrnnrq
tmedlislwqydhltatyllllakkargkpvrlrlssfscghhhhhh
Sequence, based on observed residues (ATOM records): (download)
>4bkyA (A:)
dydellkyyelhetigtggfakvklachiltgemvaikimdkntldlprikteiealknl
rhqhicqlyhvletankifmvleycpggelfdyiisqdrlseeetrvvfrqivsavayvh
sqgyahrdlkpenllfdeyhklklidfglcaslayaapeliqgkgseadvwsmgillyvl
mcgflpfdddnvmalykkimrgkydvpkwlspssilllqqmlqvdpkkrismknllnhpw
imqdynypvewqsknpfihldddcvtelsvhhrnnrqtmedlislwqydhltatylllla
kkargkpvrlr