PDB entry 4bhz

View 4bhz on RCSB PDB site
Description: Scaffold Focused Virtual Screening: Prospective Application to the Discovery of TTK Inhibitor
Class: transferase
Keywords: transferase, mitosis
Deposited on 2013-04-09, released 2013-05-22
The last revision prior to the SCOPe 2.05 freeze date was dated 2013-06-05, with a file datestamp of 2013-05-31.
Experiment type: XRAY
Resolution: 2.85 Å
R-factor: 0.1888
AEROSPACI score: 0.28 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Dual specificity protein kinase TTK
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed):
    • Uniprot P33981 (23-End)
      • expression tag (20-22)
    Domains in SCOPe 2.05: d4bhza_
  • Heterogens: 7PE, Z0B, EDO, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >4bhzA (A:)
    mhhhhhhssgvdlgtenlyfqsmsvkgriysilkqigsggsskvfqvlnekkqiyaikyv
    nleeadnqtldsyrneiaylnklqqhsdkiirlydyeitdqyiymvmecgnidlnswlkk
    kksidpwerksywknmleavhtihqhgivhsdlkpanflivdgmlklidfgianqmqpdt
    tsvvkdsqvgtvnymppeaikdmsssrengkskskispksdvwslgcilyymtygktpfq
    qiinqisklhaiidpnheiefpdipekdlqdvlkcclkrdpkqrisipellahpyvqiqt
    hpvnqmakgttee
    

    Sequence, based on observed residues (ATOM records): (download)
    >4bhzA (A:)
    qsmsvkgriysilkqigsskvfqvlnekkqiyaikyvnleeadnqtldsyrneiaylnkl
    qqhsdkiirlydyeitdqyiymvmecgnidlnswlkkkksidpwerksywknmleavhti
    hqhgivhsdlkpanflivdgmlklidfgianqqvgtvnymppeaikdispksdvwslgci
    lyymtygktpfqqiinqisklhaiidpnheiefpdipekdlqdvlkcclkrdpkqrisip
    ellahpyvqiq