PDB entry 4bhz
View 4bhz on RCSB PDB site
Description: Scaffold Focused Virtual Screening: Prospective Application to the Discovery of TTK Inhibitor
Class: transferase
Keywords: transferase, mitosis
Deposited on
2013-04-09, released
2013-05-22
The last revision prior to the SCOPe 2.05 freeze date was dated
2013-06-05, with a file datestamp of
2013-05-31.
Experiment type: XRAY
Resolution: 2.85 Å
R-factor: 0.1888
AEROSPACI score: 0.28
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Dual specificity protein kinase TTK
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d4bhza_ - Heterogens: 7PE, Z0B, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4bhzA (A:)
mhhhhhhssgvdlgtenlyfqsmsvkgriysilkqigsggsskvfqvlnekkqiyaikyv
nleeadnqtldsyrneiaylnklqqhsdkiirlydyeitdqyiymvmecgnidlnswlkk
kksidpwerksywknmleavhtihqhgivhsdlkpanflivdgmlklidfgianqmqpdt
tsvvkdsqvgtvnymppeaikdmsssrengkskskispksdvwslgcilyymtygktpfq
qiinqisklhaiidpnheiefpdipekdlqdvlkcclkrdpkqrisipellahpyvqiqt
hpvnqmakgttee
Sequence, based on observed residues (ATOM records): (download)
>4bhzA (A:)
qsmsvkgriysilkqigsskvfqvlnekkqiyaikyvnleeadnqtldsyrneiaylnkl
qqhsdkiirlydyeitdqyiymvmecgnidlnswlkkkksidpwerksywknmleavhti
hqhgivhsdlkpanflivdgmlklidfgianqqvgtvnymppeaikdispksdvwslgci
lyymtygktpfqqiinqisklhaiidpnheiefpdipekdlqdvlkcclkrdpkqrisip
ellahpyvqiq