PDB entry 4bdd
View 4bdd on RCSB PDB site
Description: Fragment-based screening identifies a new area for inhibitor binding to checkpoint kinase 2 (CHK2)
Class: transferase
Keywords: transferase, inhibitor
Deposited on
2012-10-05, released
2013-06-26
The last revision prior to the SCOPe 2.05 freeze date was dated
2013-06-26, with a file datestamp of
2013-06-21.
Experiment type: XRAY
Resolution: 2.67 Å
R-factor: 0.188
AEROSPACI score: 0.31
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: serine/threonine-protein kinase chk2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d4bdda_ - Heterogens: EDO, Z0O, NO3, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4bddA (A:)
gplgshmsvypkalrdeyimsktlgsgacgevklaferktckkvaikiiskrkfaigsar
eadpalnveteieilkklnhpciikiknffdaedyyivlelmeggelfdkvvgnkrlkea
tcklyfyqmllavqylhengiihrdlkpenvllssqeedclikitdfghskilgetslmr
tlcgtptylapevlvsvgtagynravdcwslgvilficlsgyppfsehrtqvslkdqits
gkynfipevwaevsekaldlvkkllvvdpkarftteealrhpwlqdedmkrkfqdllsee
nestalpqvlaqpstsrkrpregeaegae
Sequence, based on observed residues (ATOM records): (download)
>4bddA (A:)
msvypkalrdeyimsktlevklaferktckkvaikiisknveteieilkklnhpciikik
nffdaedyyivlelmeggelfdkvvgnkrlkeatcklyfyqmllavqylhengiihrdlk
penvllssqeedclikitdfghskiltslmrtlcgtptylapevlvsvgtagynravdcw
slgvilficlsgyppfsehrtqvslkdqitsgkynfipevwaevsekaldlvkkllvvdp
karftteealrhpwlqdedmkrkfqdllseenestalpqvl