PDB entry 4awq

View 4awq on RCSB PDB site
Description: Complex of HSP90 ATPase domain with tropane derived inhibitors
Class: chaperone
Keywords: chaperone
Deposited on 2012-06-05, released 2012-08-29
The last revision prior to the SCOPe 2.08 freeze date was dated 2017-06-28, with a file datestamp of 2017-06-23.
Experiment type: XRAY
Resolution: 1.6 Å
R-factor: N/A
AEROSPACI score: 0.44 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Heat shock protein HSP 90-alpha
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d4awqa_
  • Chain 'B':
    Compound: Heat shock protein HSP 90-alpha
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d4awqb_
  • Heterogens: 592, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >4awqA (A:)
    gsdqpmeeeevetfafqaeiaqlmsliintfysnkeiflrelisnssdaldkiryesltd
    pskldsgkelhinlipnkqdrtltivdtgigmtkadlinnlgtiaksgtkafmealqaga
    dismigqfgvgfysaylvaekvtvitkhnddeqyawessaggsftvrtdtgepmgrgtkv
    ilhlkedqteyleerrikeivkkhsqfigypitlfvekerdkevsddeae
    

    Sequence, based on observed residues (ATOM records): (download)
    >4awqA (A:)
    vetfafqaeiaqlmsliintfysnkeiflrelisnssdaldkiryesltdpskldsgkel
    hinlipnkqdrtltivdtgigmtkadlinnlgtiaksgtkafmealqdismigqfgvgfy
    saylvaekvtvitkhnddeqyawessaggsftvrtdtgepmgrgtkvilhlkedqteyle
    errikeivkkhsqfigypitlfve
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >4awqB (B:)
    gsdqpmeeeevetfafqaeiaqlmsliintfysnkeiflrelisnssdaldkiryesltd
    pskldsgkelhinlipnkqdrtltivdtgigmtkadlinnlgtiaksgtkafmealqaga
    dismigqfgvgfysaylvaekvtvitkhnddeqyawessaggsftvrtdtgepmgrgtkv
    ilhlkedqteyleerrikeivkkhsqfigypitlfvekerdkevsddeae
    

    Sequence, based on observed residues (ATOM records): (download)
    >4awqB (B:)
    vetfafqaeiaqlmsliintfysnkeiflrelisnssdaldkiryesltdpskldsgkel
    hinlipnkqdrtltivdtgigmtkadlinnlgtiaksgtkafmealqdismigqfgvgfy
    saylvaekvtvitkhnddeqyawessaggsftvrtdtgepmgrgtkvilhlkedqteyle
    errikeivkkhsqfigypitlfve