PDB entry 4aw5

View 4aw5 on RCSB PDB site
Description: Complex of the EphB4 kinase domain with an oxindole inhibitor
Class: transferase
Keywords: transferase
Deposited on 2012-05-31, released 2012-08-01
The last revision prior to the SCOPe 2.08 freeze date was dated 2012-08-01, with a file datestamp of 2012-07-27.
Experiment type: XRAY
Resolution: 2.33 Å
R-factor: 0.19439
AEROSPACI score: 0.36 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Ephrin type-B receptor 4
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d4aw5a_
  • Heterogens: 30K, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >4aw5A (A:)
    pwgsmefakeidvsyvkieevigagefgevcrgrlkapgkkescvaiktlkggyterqrr
    eflseasimgqfehpniirlegvvtnsmpvmiltefmengaldsflrlndgqftviqlvg
    mlrgiasgmrylaemsyvhrdlaarnilvnsnlvckvsdfglsrfleenssdptytsslg
    gkipirwtapeaiafrkftsasdawsygivmwevmsfgerpywdmsnqdvinaieqdyrl
    ppppdcptslhqlmldcwqkdrnarprfpqvvsaldkmirnpaslkivare
    

    Sequence, based on observed residues (ATOM records): (download)
    >4aw5A (A:)
    akeidvsyvkieevigagefgevcrgrlkapgkkescvaiktlkggyterqrreflseas
    imgqfehpniirlegvvtnsmpvmiltefmengaldsflrlndgqftviqlvgmlrgias
    gmrylaemsyvhrdlaarnilvnsnlvckvsdfgipirwtapeaiafrkftsasdawsyg
    ivmwevmsfgerpywdmsnqdvinaieqdyrlppppdcptslhqlmldcwqkdrnarprf
    pqvvsaldkmirnpaslkiva