PDB entry 4ans
View 4ans on RCSB PDB site
Description: Structure of L1196M,G1269A Double Mutant Anaplastic Lymphoma Kinase in Complex with Crizotinib
Class: transferase
Keywords: transferase
Deposited on
2012-03-22, released
2013-03-27
The last revision prior to the SCOPe 2.05 freeze date was dated
2013-03-27, with a file datestamp of
2013-03-22.
Experiment type: XRAY
Resolution: 1.85 Å
R-factor: 0.201
AEROSPACI score: 0.49
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: ALK tyrosine kinase receptor
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- Uniprot Q9UM73 (23-End)
- engineered mutation (126)
- engineered mutation (199)
Domains in SCOPe 2.05: d4ansa_ - Heterogens: VGH, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4ansA (A:)
mahhhhhhdygipttenlyfqgsnpnycfagktssisdlkevprknitlirglghgafge
vyegqvsgmpndpsplqvavktlpevcseqdeldflmealiiskfnhqnivrcigvslqs
lprfilmelmaggdlksflretrprpsqpsslamldllhvardiacgcqyleenhfihrd
iaarnclltcpgpgrvakiadfgmardiyrasyyrkggcamlpvkwmppeafmegiftsk
tdtwsfgvllweifslgympypsksnqevlefvtsggrmdppkncpgpvyrimtqcwqhq
pedrpnfaiilerieyctqdpdvintalpieygplveeeekv
Sequence, based on observed residues (ATOM records): (download)
>4ansA (A:)
npnycfagktssisdlkevprknitlirglgafgevyegqvplqvavktlpevcseqdel
dflmealiiskfnhqnivrcigvslqslprfilmelmaggdlksflretrprpsqpssla
mldllhvardiacgcqyleenhfihrdiaarnclltcpgpgrvakiadfgmardiyrggc
amlpvkwmppeafmegiftsktdtwsfgvllweifslgympypsksnqevlefvtsggrm
dppkncpgpvyrimtqcwqhqpedrpnfaiilerieyctqdpdvintalpieyg