PDB entry 4a9o
View 4a9o on RCSB PDB site
Description: N-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 5 ethyl-3-methyl-4-phenyl-1, 2-oxazole
Class: signaling protein/inhibitor
Keywords: signaling protein-inhibitor complex
Deposited on
2011-11-26, released
2012-02-08
The last revision prior to the SCOPe 2.04 freeze date was dated
2012-02-08, with a file datestamp of
2012-02-03.
Experiment type: XRAY
Resolution: 1.78 Å
R-factor: 0.17333
AEROSPACI score: 0.55
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: bromodomain containing 2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.04: d4a9oa_ - Chain 'B':
Compound: bromodomain containing 2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.04: d4a9ob_ - Chain 'C':
Compound: bromodomain containing 2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.04: d4a9oc_ - Heterogens: EDO, A9O, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4a9oA (A:)
gsshhhhhhssglvprgshmsnpkkpgrvtnqlqylhkvvmkalwkhqfawpfrqpvdav
klglpdyhkiikqpmdmgtikrrlennyywaasecmqdfntmftncyiynkptddivlma
qtlekiflqkvasmpqeeqelvvtipknshkkga
Sequence, based on observed residues (ATOM records): (download)
>4a9oA (A:)
rvtnqlqylhkvvmkalwkhqfawpfrqpvdavklglpdyhkiikqpmdmgtikrrlenn
yywaasecmqdfntmftncyiynkptddivlmaqtlekiflqkvasmpqeeqelv
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4a9oB (B:)
gsshhhhhhssglvprgshmsnpkkpgrvtnqlqylhkvvmkalwkhqfawpfrqpvdav
klglpdyhkiikqpmdmgtikrrlennyywaasecmqdfntmftncyiynkptddivlma
qtlekiflqkvasmpqeeqelvvtipknshkkga
Sequence, based on observed residues (ATOM records): (download)
>4a9oB (B:)
tnqlqylhkvvmkalwkhqfawpfrqpvdavklglpdyhkiikqpmdmgtikrrlennyy
waasecmqdfntmftncyiynkptddivlmaqtlekiflqkvasmpqe
- Chain 'C':
Sequence, based on SEQRES records: (download)
>4a9oC (C:)
gsshhhhhhssglvprgshmsnpkkpgrvtnqlqylhkvvmkalwkhqfawpfrqpvdav
klglpdyhkiikqpmdmgtikrrlennyywaasecmqdfntmftncyiynkptddivlma
qtlekiflqkvasmpqeeqelvvtipknshkkga
Sequence, based on observed residues (ATOM records): (download)
>4a9oC (C:)
tnqlqylhkvvmkalwkhqfawpfrqpvdavklglpdyhkiikqpmdmgtikrrlennyy
waasecmqdfntmftncyiynkptddivlmaqtlekiflqkvasmpq