PDB entry 4a9k
View 4a9k on RCSB PDB site
Description: BROMODOMAIN OF HUMAN CREBBP WITH N-(4-hydroxyphenyl)acetamide
Class: signaling protein
Keywords: inhibitor, histone, epigenetic reader, signaling protein
Deposited on
2011-11-26, released
2012-01-11
The last revision prior to the SCOPe 2.02 freeze date was dated
2012-02-08, with a file datestamp of
2012-02-03.
Experiment type: XRAY
Resolution: 1.81 Å
R-factor: 0.16175
AEROSPACI score: 0.54
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: creb-binding protein
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d4a9ka_ - Chain 'B':
Compound: creb-binding protein
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d4a9kb_ - Heterogens: EDO, TYL, SCN, K, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4a9kA (A:)
smrkkifkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlsti
krkldtgqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqslg
Sequence, based on observed residues (ATOM records): (download)
>4a9kA (A:)
kifkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlstikrkl
dtgqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqslg
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4a9kB (B:)
smrkkifkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlsti
krkldtgqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqslg
Sequence, based on observed residues (ATOM records): (download)
>4a9kB (B:)
fkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlstikrkldt
gqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqsl