PDB entry 4a07
View 4a07 on RCSB PDB site
Description: human pdk1 kinase domain in complex with allosteric activator ps171 bound to the pif-pocket
Class: transferase
Keywords: transferase, allosteric site
Deposited on
2011-09-08, released
2011-12-07
The last revision prior to the SCOPe 2.05 freeze date was dated
2011-12-21, with a file datestamp of
2011-12-16.
Experiment type: XRAY
Resolution: 1.85 Å
R-factor: 0.1609
AEROSPACI score: 0.38
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: 3-phosphoinositide-dependent protein kinase 1
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- Uniprot O15530 (Start-310)
- engineered mutation (239)
- engineered mutation (243)
Domains in SCOPe 2.05: d4a07a_ - Heterogens: ATP, AZ7, MG, CL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4a07A (A:)
gamdgtaaeprpgagslqhaqpppqprkkrpedfkfgkilgegsfstvvlarelatsrey
aikilekrhiikenkvpyvtrerdvmsrldhpffvklyftfqddeklyfglsyakngell
kyirkigsfdetctrfytaeivsaleylhgkgiihrdlkpenillnedmhiqitdfgtak
vlspeskqaransfvgtaqyvspellteksackssdlwalgciiyqlvaglppfragneg
lifakiikleydfpekffpkardlvekllvldatkrlgceemegygplkahpffesvtwe
nlhqqtppklt
Sequence, based on observed residues (ATOM records): (download)
>4a07A (A:)
rkkrpedfkfgkilgegsfstvvlarelatsreyaikilekrhiikenkvpyvtrerdvm
srldhpffvklyftfqddeklyfglsyakngellkyirkigsfdetctrfytaeivsale
ylhgkgiihrdlkpenillnedmhiqitdfgtakvlspeskqaransfvgtaqyvspell
teksackssdlwalgciiyqlvaglppfragneglifakiikleydfpekffpkardlve
kllvldatkrlgceemegygplkahpffesvtwenlhqqtppklt