PDB entry 3wq9
View 3wq9 on RCSB PDB site
Description: Crystal structure of Hsp90-alpha N-terminal domain in complex with 2-(4-Hydroxy-cyclohexylamino)-4-[5-(4-phenyl-imidazol-1-yl)-isoquinolin-1-yl]-benzamide
Class: chaperone
Keywords: HYDROLASE, ATP Binding, CHAPERONE
Deposited on
2014-01-23, released
2015-02-25
The last revision prior to the SCOPe 2.07 freeze date was dated
2015-02-25, with a file datestamp of
2015-02-20.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: 0.217
AEROSPACI score: 0.4
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Heat shock protein HSP 90-alpha
Species: Homo sapiens [TaxId:9606]
Gene: HSP90AA1, HSP90A, HSPC1, HSPCA
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d3wq9a_ - Heterogens: YUK, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3wq9A (A:)
hmpeetqtqdqpmeeeevetfafqaeiaqlmsliintfysnkeiflrelisnssdaldki
ryesltdpskldsgkelhinlipnkqdrtltivdtgigmtkadlinnlgtiaksgtkafm
ealqagadismigqfgvgfysaylvaekvtvitkhnddeqyawessaggsftvrtdtgep
mgrgtkvilhlkedqteyleerrikeivkkhsqfigypitlfvekerdkevsddeae
Sequence, based on observed residues (ATOM records): (download)
>3wq9A (A:)
evetfafqaeiaqlmsliintfysnkeiflrelisnssdaldkiryesltdpskldsgke
lhinlipnkqdrtltivdtgigmtkadlinnlgtiaksgtkafmealqagadismigqfg
vgfysaylvaekvtvitkhnddeqyawessaggsftvrtdtgepmgrgtkvilhlkedqt
eyleerrikeivkkhsqfigypitlfveker