PDB entry 3wbl
View 3wbl on RCSB PDB site
Description: Crystal structure of CDK2 in complex with pyrazolopyrimidine inhibitor
Class: transferase/transferase inhibitor
Keywords: Binding Sites, Tumor, Cyclin-Dependent Kinase 2, Drug Design, MAP Kinase Kinase 2, MK2, Protein Kinase Inhibitors, Pyrazoles, Pyrimidines, Structure-Activity Relationship, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2013-05-20, released
2013-10-30
The last revision prior to the SCOPe 2.06 freeze date was dated
2013-10-30, with a file datestamp of
2013-10-25.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.192
AEROSPACI score: 0.37
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cyclin-dependent kinase 2
Species: Homo sapiens [TaxId:9606]
Gene: CDK2, CDKN2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3wbla_ - Heterogens: ACT, PDY, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3wblA (A:)
menfqkvekigegtygvvykarnkltgevvalkkirldtetegvpstaireisllkelnh
pnivklldvihtenklylvfeflhqdlkkfmdasaltgiplpliksylfqllqglafchs
hrvlhrdlkpqnllintegaikladfglarafgvpvrtythevvtlwyrapeillgckyy
stavdiwslgcifaemvtrralfpgdseidqlfrifrtlgtpdevvwpgvtsmpdykpsf
pkwarqdfskvvppldedgrsllsqmlhydpnkrisakaalahpffqdvtkpvphlrl
Sequence, based on observed residues (ATOM records): (download)
>3wblA (A:)
menfqkvekigegtygvvykarnktgevvalkkirlgvpstaireisllkelnhpnivkl
ldvihtenklylvfeflhqdlkkfmdasaltgiplpliksylfqllqglafchshrvlhr
dlkpqnllintegaikladfglarafgvvtlwyrapeillgckyystavdiwslgcifae
mvtrralfpgdseidqlfrifrtlgtpdevvwpgvtsmpdykpsfpkwarqdfskvvppl
dedgrsllsqmlhydpnkrisakaalahpffqdvtkpvphlrl