PDB entry 3w87
View 3w87 on RCSB PDB site
Description: Structure of Trypanosoma cruzi dihydroorotate dehydrogenase in complex with SH-1-103
Class: oxidoreductase/oxidoreductase inhibitor
Keywords: Rossmann Fold, Oxidoreductase, Dihydroorotate/orotate and fumarate/succinate binding, Cytosol, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR complex
Deposited on
2013-03-12, released
2014-04-09
The last revision prior to the SCOPe 2.06 freeze date was dated
2014-04-09, with a file datestamp of
2014-04-04.
Experiment type: XRAY
Resolution: 1.43 Å
R-factor: 0.155
AEROSPACI score: 0.61
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Dihydroorotate dehydrogenase (fumarate)
Species: Trypanosoma cruzi [TaxId:353153]
Gene: PyrD
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3w87a1, d3w87a2 - Chain 'B':
Compound: Dihydroorotate dehydrogenase (fumarate)
Species: Trypanosoma cruzi [TaxId:353153]
Gene: PyrD
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3w87b1, d3w87b2 - Heterogens: W87, GOL, CAC, FMN, EDO, PEG, NCO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>3w87A (A:)
smclklnlldhvfanpfmnaagvlcsteedlrcmtasssgalvsksctsaprdgnpepry
mafplgsinsmglpnlgfdfylkyasdlhdyskkplflsisglsveenvamvrrlapvaq
ekgvllelnlscpnvpgkpqvaydfeamrtylqqvslayglpfgvkmppyfdiahfdtaa
avlnefplvkfvtcvnsvgnglvidaesesvvikpkqgfgglggkyilptalanvnafyr
rcpdklvfgcggvysgedaflhilagasmvqvgtalqeegpgiftrledelleimarkgy
rtleefrgrvktie
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>3w87B (B:)
smclklnlldhvfanpfmnaagvlcsteedlrcmtasssgalvsksctsaprdgnpepry
mafplgsinsmglpnlgfdfylkyasdlhdyskkplflsisglsveenvamvrrlapvaq
ekgvllelnlscpnvpgkpqvaydfeamrtylqqvslayglpfgvkmppyfdiahfdtaa
avlnefplvkfvtcvnsvgnglvidaesesvvikpkqgfgglggkyilptalanvnafyr
rcpdklvfgcggvysgedaflhilagasmvqvgtalqeegpgiftrledelleimarkgy
rtleefrgrvktie