PDB entry 3w55
View 3w55 on RCSB PDB site
Description: The structure of ERK2 in complex with FR148083
Class: transferase/transferase inhibitor
Keywords: PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2013-01-21, released
2013-02-06
The last revision prior to the SCOPe 2.04 freeze date was dated
2013-02-06, with a file datestamp of
2013-02-01.
Experiment type: XRAY
Resolution: 3 Å
R-factor: 0.262
AEROSPACI score: 0.14
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 1
Species: Homo sapiens [TaxId:9606]
Gene: MAPK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.04: d3w55a_ - Heterogens: 1FM, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3w55A (A:)
gdlgsdelmaaaaaagagpemvrgqvfdvgprytnlsyigegaygmvcsaydnvnkvrva
ikkispfehqtycqrtlreikillrfrheniigindiiraptieqmkdvyivqdlmetdl
ykllktqhlsndhicyflyqilrglkyihsanvlhrdlkpsnlllnttcdlkicdfglar
vadpdhdhtgflteyvatrwyrapeimlnskgytksidiwsvgcilaemlsnrpifpgkh
yldqlnhilgilgspsqedlnciinlkarnyllslphknkvpwnrlfpnadskaldlldk
mltfnphkrieveqalahpyleqyydpsdepiaeapfkfdmelddlpkeklkelifeeta
rfqpgyrs
Sequence, based on observed residues (ATOM records): (download)
>3w55A (A:)
pemvrgqvfdvgprytnlsyigegaygmvcsaydnvnkvrvaikkispfehqtycqrtlr
eikillrfrheniigindiiraptieqmkdvyivqdlmetdlykllktqhlsndhicyfl
yqilrglkyihsanvlhrdlkpsnlllnttcdlkicdfglarvadvatrwyrapeimlns
kgytksidiwsvgcilaemlsnrpifpgkhyldqlnhilgilgspsqedlnciinlkarn
yllslphknkvpwnrlfpnadskaldlldkmltfnphkrieveqalahpyleqyydpsde
piaeapfkfdmelddlpkeklkelifeetarfqpg