PDB entry 3vqc
View 3vqc on RCSB PDB site
Description: HIV-1 IN core domain in complex with (5-METHYL-3-PHENYL-1,2-OXAZOL-4-YL)METHANOL
Class: transferase/transferase inhibitor
Keywords: rnaseH, DNA binding, DNA cleavage, DNA integration, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2012-03-21, released
2013-01-30
The last revision prior to the SCOPe 2.07 freeze date was dated
2013-01-30, with a file datestamp of
2013-01-25.
Experiment type: XRAY
Resolution: 2.3 Å
R-factor: 0.222
AEROSPACI score: 0.33
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Pol polyprotein
Species: Human immunodeficiency virus 1 [TaxId:11676]
Gene: pol
Database cross-references and differences (RAF-indexed):
- Uniprot Q72498
- engineered mutation (76)
- engineered mutation (84)
- engineered mutation (130)
Domains in SCOPe 2.07: d3vqca_ - Chain 'B':
Compound: Pol polyprotein
Species: Human immunodeficiency virus 1 [TaxId:11676]
Gene: pol
Database cross-references and differences (RAF-indexed):
- Uniprot Q72498
- engineered mutation (76)
- engineered mutation (130)
Domains in SCOPe 2.07: d3vqcb_ - Heterogens: CD, SO4, MPK, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3vqcA (A:)
dsspgiwqldcthlegkvilvavhvasgyieaevipaetgqetayfllklagrwpvktvh
tdngsnftsttvkaacdwagikqedgipynpqsqgviesmnkelkkiigqvrdqaehlkt
avqmavfihnhkrkggiggysagerivdiiatdiqtke
Sequence, based on observed residues (ATOM records): (download)
>3vqcA (A:)
spgiwqldcthlegkvilvavhvasgyieaevipaetgqetayfllklagrwpvktvhtd
ngsnftsttvkaacdwagikqedgipsmnkelkkiigqvrdqaehlktavqmavfihnhk
rkggiggysagerivdiiatd
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3vqcB (B:)
dsspgiwqldcthlegkvilvavhvasgyieaevipaetgqetayfllklagrwpvktvh
tdngsnftsttvkaacdwagikqedgipynpqsqgviesmnkelkkiigqvrdqaehlkt
avqmavfihnhkrkggiggysagerivdiiatdiqtke
Sequence, based on observed residues (ATOM records): (download)
>3vqcB (B:)
spgiwqldcthlegkvilvavhvasgyieaevipaetgqetayfllklagrwpvktvhtd
ngsnftsttvkaacdwagikqesmnkelkkiigqvrdqaehlktavqmavfihnhkrkgg
iggysagerivdiiatdi